# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA288470 | 4-(dimethylamino)antipyrine | AC50 | > | 30 | uM | ALA5291731 | Summarised AC50 (mean value for measurements with a relation sign "="; largest value for measurements with relation sign ">") | nM | Homo sapiens | ||
2. | ALA288470 | 4-(dimethylamino)antipyrine | AC50 | > | 30 | uM | ALA5291887 | Summarised AC50 (mean value for measurements with a relation sign "="; largest value for measurements with relation sign ">") | nM | Homo sapiens | ||
3. | ALA288470 | 4-(dimethylamino)antipyrine | LogD7.4 | 0.78 | ALA3301363 | |||||||
4. | ALA288470 | 4-(dimethylamino)antipyrine | CLint | 3.47 | microL/min/1E6 cells | ALA3301372 | uL.min-1.(10^6cells)-1 | |||||
5. | ALA288470 | 4-(dimethylamino)antipyrine | AC50 | 0.631 | uM | ALA3562146 | inactive | nM | ||||
6. | ALA288470 | 4-(dimethylamino)antipyrine | AC50 | 0.631 | uM | ALA3562136 | inactive | nM | ||||
7. | ALA288470 | 4-(dimethylamino)antipyrine | Ac50 | 0.631 | uM | ALA3562152 | inactive | uM | ||||
8. | ALA288470 | 4-(dimethylamino)antipyrine | Ac50 | 0.631 | uM | ALA3561990 | inactive | uM | ||||
9. | ALA288470 | 4-(dimethylamino)antipyrine | Ac50 | 0.631 | uM | ALA3562064 | inactive | uM | ||||
10. | ALA288470 | 4-(dimethylamino)antipyrine | AC50 | 0.631 | uM | ALA3562119 | inactive | nM | ||||
11. | ALA288470 | 4-(dimethylamino)antipyrine | CL | 0 | ALA3534907 | Not determined | ||||||
12. | ALA288470 | 4-(dimethylamino)antipyrine | INH | < | 10 | % | ALA3534886 | % | Homo sapiens | |||
13. | ALA288470 | 4-(dimethylamino)antipyrine | INH | < | 10 | % | ALA3534885 | % | Homo sapiens | |||
14. | ALA288470 | 4-(dimethylamino)antipyrine | INH | < | 10 | % | ALA3534884 | % | Homo sapiens | |||
15. | ALA288470 | 4-(dimethylamino)antipyrine | logD | = | 0.63 | ALA3533246 | ||||||
16. | ALA288470 | 4-(dimethylamino)antipyrine | PB | = | 30.9 | pmol | ALA3534888 | pmol | Homo sapiens | |||
17. | ALA288470 | 4-(dimethylamino)antipyrine | logPapp | = | -4.44 | ALA3533248 | ||||||
18. | ALA288470 | 4-(dimethylamino)antipyrine | F | = | 100 | % | ALA3533250 | % | Homo sapiens | |||
19. | ALA288470 | 4-(dimethylamino)antipyrine | INH | < | 10 | % | ALA3534890 | % | Homo sapiens | |||
20. | ALA288470 | 4-(dimethylamino)antipyrine | INH | < | 10 | % | ALA3534883 | % | Homo sapiens |