| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA601906 | 4t | F | = | 31 | % | ALA1070732 | % | Canis lupus familiaris | |||
| 2. | ALA601906 | 4t | t1/2 | = | 0.8 | hr | ALA1070730 | hr | Canis lupus familiaris | |||
| 3. | ALA601906 | 4t | Vdss | = | 0.22 | L/Kg | ALA1070728 | L.kg-1 | Canis lupus familiaris | |||
| 4. | ALA601906 | 4t | CL | = | 3 | ml/min.kg | ALA1070726 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 5. | ALA601906 | 4t | Stability | 0 | ALA1070707 | Stable | % | |||||
| 6. | ALA601906 | 4t | Stability | 0 | ALA1070706 | Stable | % | |||||
| 7. | ALA601906 | 4t | Activity | 0 | ALA1070713 | Non-toxic | Rattus norvegicus | |||||
| 8. | ALA601906 | 4t | F | = | 89 | % | ALA1070711 | % | Rattus norvegicus | |||
| 9. | ALA601906 | 4t | t1/2eff | = | 1.5 | hr | ALA1070710 | hr | Rattus norvegicus | |||
| 10. | ALA601906 | 4t | Vdss | = | 0.7 | L/Kg | ALA1070709 | L.kg-1 | Rattus norvegicus | |||
| 11. | ALA601906 | 4t | CL | = | 5 | ml/min.kg | ALA1070708 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 12. | ALA601906 | 4t | Ki | = | 2.1 | nM | ALA1064501 | 8.68 | nM | Homo sapiens | ||
| 13. | ALA601906 | 4t | IC50 | = | 0.36 | uM | ALA1064502 | 6.44 | nM | |||
| 14. | ALA601906 | 4t | FC | = | 0.54 | ALA1070705 | ||||||
| 15. | ALA601906 | 4t | IC50 | > | 90 | uM | ALA1070712 | nM | Homo sapiens | |||
| 16. | ALA601906 | 4t | Activity | 0 | ALA1070721 | Not Active | Homo sapiens | |||||
| 17. | ALA601906 | 4t | IC50 | = | 0.255 | uM | ALA1070723 | 6.59 | nM | |||
| 18. | ALA601906 | 4t | Ki | = | 6.3 | nM | ALA1070724 | 8.20 | nM | Homo sapiens | ||
| 19. | ALA601906 | 4t | solubility | = | 921 | uM | ALA1070715 | nM | ||||
| 20. | ALA601906 | 4t | solubility | = | 195 | uM | ALA1070716 | nM |
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