| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA599217 | 21 | Ratio IC50 | = | 12 | ALA1116629 | ||||||
| 2. | ALA599217 | 21 | IC50 | = | 1.84 | uM | ALA1116628 | 5.74 | nM | |||
| 3. | ALA599217 | 21 | IC50 | = | 0.15 | uM | ALA1104120 | 6.82 | nM | Rattus norvegicus | ||
| 4. | ALA599217 | 21 | F | = | 22 | % | ALA1071415 | % | Rattus norvegicus | |||
| 5. | ALA599217 | 21 | t1/2 | = | 6 | hr | ALA1071414 | hr | Rattus norvegicus | |||
| 6. | ALA599217 | 21 | AUC | = | 2785 | nM.hr | ALA1071413 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 7. | ALA599217 | 21 | Tmax | = | 2 | hr | ALA1071412 | hr | Rattus norvegicus | |||
| 8. | ALA599217 | 21 | IC50 | = | 0.15 | uM | ALA1068015 | 6.82 | nM | Homo sapiens | ||
| 9. | ALA599217 | 21 | IC50 | = | 1.84 | uM | ALA1068016 | 5.74 | nM | Homo sapiens | ||
| 10. | ALA599217 | 21 | IC50 | = | 3.5 | uM | ALA1068017 | 5.46 | nM | Homo sapiens | ||
| 11. | ALA599217 | 21 | solubility | = | 0.38 | ug ml-1 | ALA1068018 | ug.mL-1 | ||||
| 12. | ALA599217 | 21 | Activity | = | 80.9 | % | ALA1071406 | % | Rattus norvegicus | |||
| 13. | ALA599217 | 21 | Activity | = | 97.9 | % | ALA1071407 | % | Rattus norvegicus | |||
| 14. | ALA599217 | 21 | Cmax | = | 2933 | nM | ALA1071408 | nM | Rattus norvegicus | |||
| 15. | ALA599217 | 21 | AUC | = | 2499 | nM.hr | ALA1071409 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 16. | ALA599217 | 21 | t1/2 | = | 11 | hr | ALA1071410 | hr | Rattus norvegicus | |||
| 17. | ALA599217 | 21 | Cmax | = | 292 | nM | ALA1071411 | nM | Rattus norvegicus |
The page will load shortly, Thanks for your patience!