# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1086654 | 4 | Activity | 0 | ALA4256557 | Toxic | Mus musculus | |||||
2. | ALA1086654 | 4 | Activity | 0 | ALA4256556 | Toxic | Mus musculus | |||||
3. | ALA1086654 | 4 | Activity | 0 | ALA4256555 | Toxic | Mus musculus | |||||
4. | ALA1086654 | 4 | LD50 | > | 10 | mg kg-1 | ALA4256545 | mg.kg-1 | Mus musculus | |||
5. | ALA1086654 | 4 | Imax | 0 | ALA4256540 | Not Determined | Rattus norvegicus | |||||
6. | ALA1086654 | 4 | EC50 | 0 | ALA4256539 | Not Determined | Rattus norvegicus | |||||
7. | ALA1086654 | 4 | Imax | = | 1.02 | % | ALA4256538 | % | Rattus norvegicus | |||
8. | ALA1086654 | 4 | EC50 | = | 21 | uM | ALA4256537 | 4.68 | nM | Rattus norvegicus | ||
9. | ALA1086654 | 4 | Imax | = | 0.43 | % | ALA4256536 | % | Rattus norvegicus | |||
10. | ALA1086654 | 4 | EC50 | = | 0.045 | uM | ALA4256535 | 7.35 | nM | Rattus norvegicus | ||
11. | ALA1086654 | 4 | Imax | 0 | ALA4256534 | Not Determined | Rattus norvegicus | |||||
12. | ALA1086654 | 4 | EC50 | 0 | ALA4256533 | Not Determined | Rattus norvegicus | |||||
13. | ALA1086654 | 4 | Ratio EC50 | = | 0.49 | ALA4256532 | ||||||
14. | ALA1086654 | 4 | Ki | = | 390 | nM | ALA4256520 | 6.41 | nM | Homo sapiens | ||
15. | ALA1086654 | 4 | Ki | = | 12 | nM | ALA4256521 | 7.92 | nM | Homo sapiens | ||
16. | ALA1086654 | 4 | Ki | = | 130 | nM | ALA4256522 | 6.89 | nM | Homo sapiens | ||
17. | ALA1086654 | 4 | Ratio Ki | = | 33 | ALA4256523 | ||||||
18. | ALA1086654 | 4 | Ki | = | 29 | nM | ALA4256526 | 7.54 | nM | Rattus norvegicus | ||
19. | ALA1086654 | 4 | EC50 | = | 27 | uM | ALA4256528 | 4.57 | nM | Rattus norvegicus | ||
20. | ALA1086654 | 4 | Emax | = | 53 | % | ALA4256529 | % | Rattus norvegicus |