# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1095040 | 37 | IC50 | = | 0.08 | uM | ALA1111594 | 7.10 | nM | Homo sapiens | ||
2. | ALA1095040 | 37 | INH | = | 24 | % | ALA1111587 | % | Homo sapiens | |||
3. | ALA1095040 | 37 | IC50 | > | 10 | uM | ALA1111586 | nM | Homo sapiens | |||
4. | ALA1095040 | 37 | IC50 | > | 10 | uM | ALA1111585 | nM | Homo sapiens | |||
5. | ALA1095040 | 37 | IC50 | > | 10 | uM | ALA1111584 | nM | Homo sapiens | |||
6. | ALA1095040 | 37 | INH | = | 0.006 | uM | ALA1111575 | uM | Homo sapiens | |||
7. | ALA1095040 | 37 | solubility | < | 20 | mg/ml | ALA1111576 | ug.mL-1 | ||||
8. | ALA1095040 | 37 | logD | = | 3.7 | ALA1111577 | ||||||
9. | ALA1095040 | 37 | Activity | = | 99.4 | % | ALA1111578 | % | Homo sapiens | |||
10. | ALA1095040 | 37 | Activity | = | 91 | % | ALA1111579 | % | ||||
11. | ALA1095040 | 37 | Activity | = | 40 | % | ALA1111580 | % | ||||
12. | ALA1095040 | 37 | permeability | = | 3.9 | % | ALA1111581 | % | Homo sapiens | |||
13. | ALA1095040 | 37 | IC50 | < | 0.4 | uM | ALA1111582 | nM | Homo sapiens | |||
14. | ALA1095040 | 37 | IC50 | > | 10 | uM | ALA1111583 | nM | Homo sapiens | |||
15. | ALA1095040 | 37 | IC50 | = | 2500 | nM | ALA1113302 | 5.60 | nM | Homo sapiens | ||
16. | ALA1095040 | 37 | IC50 | = | 100 | nM | ALA1113301 | 7.00 | nM | Homo sapiens | ||
17. | ALA1095040 | 37 | IC50 | = | 400 | nM | ALA1113299 | 6.40 | nM | Rattus norvegicus | ||
18. | ALA1095040 | 37 | INH | = | 93 | % | ALA1113277 | % | Homo sapiens | |||
19. | ALA1095040 | 37 | INH | = | 95 | % | ALA1113276 | % | Homo sapiens | |||
20. | ALA1095040 | 37 | INH | = | 72 | % | ALA1113297 | % | Homo sapiens |