# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1078675 | 3a | Ki | = | 6 | nM | ALA5244929 | 8.22 | nM | Trypanosoma brucei rhodesiense | ||
2. | ALA1078675 | 3a | INH | < | 5 | % | ALA1109343 | % | Trypanosoma cruzi | |||
3. | ALA1078675 | 3a | IC50 | > | 100 | uM | ALA1109346 | nM | Homo sapiens | |||
4. | ALA1078675 | 3a | GI50 | > | 100 | uM | ALA1109345 | nM | Trypanosoma brucei brucei | |||
5. | ALA1078675 | 3a | IC50 | > | 100 | uM | ALA1109344 | nM | Trypanosoma brucei | |||
6. | ALA1078675 | 3a | Kinact | = | 0.002 | /s | ALA1109342 | /s | Trypanosoma brucei rhodesiense | |||
7. | ALA1078675 | 3a | Ki(app) | = | 0.32 | uM | ALA1109342 | 6.50 | nM | Trypanosoma brucei rhodesiense | ||
8. | ALA1078675 | 3a | IC50 | < | 0.006 | uM | ALA1109342 | nM | Trypanosoma brucei rhodesiense | |||
9. | ALA1078675 | 3a | IC50 | = | 10 | uM | ALA1109341 | 5.00 | nM | Trypanosoma cruzi |