| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1080412 | 43 | CL | = | 13 | ml/min.kg | ALA1111385 | mL.min-1.kg-1 | ||||
| 2. | ALA1080412 | 43 | Ratio | 0 | ALA1111379 | Not Determined | ||||||
| 3. | ALA1080412 | 43 | F | = | 87 | % | ALA1111378 | % | Rattus norvegicus | |||
| 4. | ALA1080412 | 43 | Vdss | = | 0.3 | L/Kg | ALA1111377 | L.kg-1 | Rattus norvegicus | |||
| 5. | ALA1080412 | 43 | CL | = | 3.8 | ml/min.kg | ALA1111376 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 6. | ALA1080412 | 43 | t1/2 | = | 0.9 | hr | ALA1111375 | hr | Rattus norvegicus | |||
| 7. | ALA1080412 | 43 | CL | = | 3 | ml/min.kg | ALA1111374 | mL.min-1.kg-1 | ||||
| 8. | ALA1080412 | 43 | permeability | = | 6.3 | 10'-6 cm/s | ALA1111373 | 10'-6 cm/s | ||||
| 9. | ALA1080412 | 43 | logD | = | 2 | ALA1111372 | ||||||
| 10. | ALA1080412 | 43 | solubility | = | 58 | mg/L | ALA1111371 | ug.mL-1 | ||||
| 11. | ALA1080412 | 43 | Efficacy | = | 21 | % | ALA1111370 | % | Rattus norvegicus | |||
| 12. | ALA1080412 | 43 | Efficacy | = | 2 | % | ALA1111369 | % | Rattus norvegicus | |||
| 13. | ALA1080412 | 43 | Efficacy | = | -20 | % | ALA1111368 | % | Rattus norvegicus | |||
| 14. | ALA1080412 | 43 | Ki | = | 48 | nM | ALA1111367 | 7.32 | nM | Homo sapiens | ||
| 15. | ALA1080412 | 43 | Ki | = | 81 | nM | ALA1111366 | 7.09 | nM | Homo sapiens | ||
| 16. | ALA1080412 | 43 | Ki | = | 53 | nM | ALA1111365 | 7.28 | nM | Homo sapiens | ||
| 17. | ALA1080412 | 43 | Efficacy | = | -18 | % | ALA1111359 | % | Rattus norvegicus | |||
| 18. | ALA1080412 | 43 | Ki | = | 5.6 | nM | ALA1111355 | 8.25 | nM | Homo sapiens |
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