# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1089116 | 1 | Activity | = | 7.7 | min | ALA1104790 | min | Homo sapiens | |||
2. | ALA1089116 | 1 | IC50 | < | 0.1 | uM | ALA1108285 | nM | Homo sapiens | |||
3. | ALA1089116 | 1 | IC50 | < | 0.1 | uM | ALA1108284 | nM | Homo sapiens | |||
4. | ALA1089116 | 1 | Vdss | = | 1.7 | L/Kg | ALA1108283 | L.kg-1 | Rattus norvegicus | |||
5. | ALA1089116 | 1 | t1/2 | = | 12 | min | ALA1108282 | hr | Rattus norvegicus | |||
6. | ALA1089116 | 1 | CL | = | 128 | ml/min.Kg | ALA1108281 | mL.min-1.kg-1 | Rattus norvegicus | |||
7. | ALA1089116 | 1 | IC50 | = | 398 | nM | ALA1108263 | 6.40 | nM | Homo sapiens | ||
8. | ALA1089116 | 1 | IC50 | = | 316 | nM | ALA1104805 | 6.50 | nM | Homo sapiens | ||
9. | ALA1089116 | 1 | IC50 | = | 398 | nM | ALA1108262 | 6.40 | nM | Homo sapiens | ||
10. | ALA1089116 | 1 | IC50 | = | 158 | nM | ALA1108261 | 6.80 | nM | Homo sapiens | ||
11. | ALA1089116 | 1 | Time | = | 7.7 | min | ALA1108275 | hr | Homo sapiens | |||
12. | ALA1089116 | 1 | EC50 | = | 79 | nM | ALA1104794 | 7.10 | nM | Homo sapiens | ||
13. | ALA1089116 | 1 | IC50 | = | 631 | nM | ALA1104791 | 6.20 | nM | Homo sapiens | ||
14. | ALA1089116 | 1 | IC50 | = | 2 | nM | ALA1104788 | 8.70 | nM | Homo sapiens | ||
15. | ALA1089116 | 1 | Selectivity ratio | > | 70 | ALA1105647 | ||||||
16. | ALA1089116 | 1 | Selectivity ratio | > | 70 | ALA1105646 | ||||||
17. | ALA1089116 | 1 | Selectivity ratio | > | 70 | ALA1105645 | ||||||
18. | ALA1089116 | 1 | Selectivity ratio | > | 70 | ALA1105644 | ||||||
19. | ALA1089116 | 1 | Selectivity ratio | > | 70 | ALA1105643 | ||||||
20. | ALA1089116 | 1 | Selectivity ratio | > | 70 | ALA1105642 |