| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1096256 | 1 | IC50 | = | 2.3 | uM | ALA3136328 | 5.64 | nM | Homo sapiens | ||
| 2. | ALA1096256 | 1 | IC50 | = | 0.14 | uM | ALA3136327 | 6.85 | nM | Homo sapiens | ||
| 3. | ALA1096256 | 1 | IC50 | = | 2.8 | uM | ALA3136326 | 5.55 | nM | |||
| 4. | ALA1096256 | 1 | AUC | = | 53.22 | uM.hr | ALA3136325 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 5. | ALA1096256 | 1 | AUC | = | 3.41 | uM.hr | ALA3136324 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 6. | ALA1096256 | 1 | Ratio AUC | = | 6.4 | % | ALA3136323 | % | Rattus norvegicus | |||
| 7. | ALA1096256 | 1 | PB | 0 | ALA3378726 | Not Active | % | Homo sapiens | ||||
| 8. | ALA1096256 | 1 | PB | 0 | ALA3378725 | Not Active | % | Mus musculus | ||||
| 9. | ALA1096256 | 1 | PPB | 0 | ALA3378724 | Not Active | % | Mus musculus | ||||
| 10. | ALA1096256 | 1 | Stability | 0 | ALA3378720 | Stable | % | Homo sapiens | ||||
| 11. | ALA1096256 | 1 | Stability | 0 | ALA3378719 | Stable | % | Mus musculus | ||||
| 12. | ALA1096256 | 1 | Stability | 0 | ALA3378718 | Stable | % | Mus musculus | ||||
| 13. | ALA1096256 | 1 | Stability | 0 | ALA3378717 | Stable | % | Homo sapiens | ||||
| 14. | ALA1096256 | 1 | EC50 | 0 | ALA3378134 | Not Determined | Homo sapiens | |||||
| 15. | ALA1096256 | 1 | EC50 | 0 | ALA3378133 | Not Determined | ||||||
| 16. | ALA1096256 | 1 | EC50 | 0 | ALA3378131 | Not Determined | ||||||
| 17. | ALA1096256 | 1 | Drug recovery | = | 65 | % | ALA3378729 | % | Homo sapiens | |||
| 18. | ALA1096256 | 1 | Drug recovery | = | 65 | % | ALA3378728 | % | Mus musculus | |||
| 19. | ALA1096256 | 1 | Drug recovery | = | 65 | % | ALA3378727 | % | Mus musculus | |||
| 20. | ALA1096256 | 1 | IC50 | = | 60 | nM | ALA3378723 | 7.22 | nM |
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