| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1083358 | 10 | IC50 | = | 27 | nM | ALA3771998 | 7.57 | nM | Homo sapiens | ||
| 2. | ALA1083358 | 10 | IC50 | = | 27 | nM | ALA3771845 | 7.57 | nM | Homo sapiens | ||
| 3. | ALA1083358 | 10 | Activity | = | 90 | % | ALA3625769 | % | Rattus norvegicus | |||
| 4. | ALA1083358 | 10 | Activity | 0 | ALA3625767 | Active | Rattus norvegicus | |||||
| 5. | ALA1083358 | 10 | Activity | 0 | ALA3625766 | Active | Rattus norvegicus | |||||
| 6. | ALA1083358 | 10 | Activity | 0 | ALA3625765 | Active | Rattus norvegicus | |||||
| 7. | ALA1083358 | 10 | Cmax | = | 2 | uM | ALA3625763 | nM | Rattus norvegicus | |||
| 8. | ALA1083358 | 10 | Tmax | = | 1.3 | hr | ALA3625762 | hr | Rattus norvegicus | |||
| 9. | ALA1083358 | 10 | AUC | = | 4.5 | uM.hr | ALA3625761 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 10. | ALA1083358 | 10 | Ki | = | 0.2 | nM | ALA3625143 | 9.70 | nM | |||
| 11. | ALA1083358 | 10 | Ki | = | 1.8 | nM | ALA3625144 | 8.74 | nM | Homo sapiens | ||
| 12. | ALA1083358 | 10 | Ratio | = | 2.5 | ALA3625149 | Rattus norvegicus | |||||
| 13. | ALA1083358 | 10 | Ratio | = | 3.8 | ALA3625148 | Homo sapiens | |||||
| 14. | ALA1083358 | 10 | CL | = | 3 | ml/min.kg | ALA3625147 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 15. | ALA1083358 | 10 | IC50 | = | 27 | nM | ALA3625146 | 7.57 | nM | Homo sapiens | ||
| 16. | ALA1083358 | 10 | IC50 | = | 27 | nM | ALA3625145 | 7.57 | nM | |||
| 17. | ALA1083358 | 10 | Drug metabolism | 0 | ALA3267711 | metabolite_detected | Homo sapiens | |||||
| 18. | ALA1083358 | 10 | Drug metabolism | 0 | ALA3267710 | metabolite_detected | Rattus norvegicus | |||||
| 19. | ALA1083358 | 10 | Time | = | 7 | min | ALA3267705 | hr | Rattus norvegicus | |||
| 20. | ALA1083358 | 10 | Time | = | 41 | min | ALA3267704 | hr | Rattus norvegicus |
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