# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1083675 | 12 | IC50 | = | 4.8 | nM | ALA1120160 | 8.32 | nM | Homo sapiens | ||
2. | ALA1083675 | 12 | IC50 | = | 58 | nM | ALA1120161 | 7.24 | nM | Rattus norvegicus | ||
3. | ALA1083675 | 12 | Cmax | = | 9.2 | ug ml-1 | ALA1120162 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
4. | ALA1083675 | 12 | AUC | = | 103.9 | microg.hr/mL | ALA1120163 | ng.hr.mL-1 | Rattus norvegicus | |||
5. | ALA1083675 | 12 | Selectivity ratio | = | 2083 | ALA1119725 | ||||||
6. | ALA1083675 | 12 | Selectivity ratio | > | 4167 | ALA1119724 | ||||||
7. | ALA1083675 | 12 | Selectivity ratio | > | 4167 | ALA1119723 | ||||||
8. | ALA1083675 | 12 | IC50 | = | 4.8 | nM | ALA1119720 | 8.32 | nM | Homo sapiens |