# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PF-4618433 | 63, PF-4618433 | CLH | = | 109 | ml/min.kg | ALA2209548 | mL.min-1.kg-1 | Homo sapiens | |||
2. | PF-4618433 | 63, PF-4618433 | IC50 | > | 10000 | nM | ALA2209546 | nM | Homo sapiens | |||
3. | PF-4618433 | 63, PF-4618433 | IC50 | = | 190 | nM | ALA2209549 | 6.72 | nM | Mus musculus | ||
4. | PF-4618433 | 63, PF-4618433 | IC50 | = | 637 | nM | ALA2209550 | 6.20 | nM | Homo sapiens | ||
5. | PF-4618433 | 63, PF-4618433 | INH | = | 16 | % | ALA2209547 | % | Homo sapiens | |||
6. | PF-4618433 | 63, PF-4618433 | IC50 | = | 637 | nM | ALA1117898 | 6.20 | nM | Homo sapiens |