# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PF-562271 | PF-562271 | Kd | = | 88 | uM | ALA5223598 | 4.06 | nM | Homo sapiens | ||
2. | PF-562271 | PF-562271 | LogD7.4 | 2.63 | ALA3301363 | |||||||
3. | PF-562271 | PF-562271 | Kd | = | 88 | uM | ALA4052313 | 4.06 | nM | Homo sapiens | ||
4. | PF-562271 | PF-562271 | Potency | 1.482 | uM | ALA3562002 | active | nM | ||||
5. | PF-562271 | PF-562271 | Potency | 2.957 | uM | ALA3562034 | active | nM | ||||
6. | PF-562271 | PF-562271 | Potency | 0.132 | uM | ALA3562018 | active | nM | ||||
7. | PF-562271 | PF-562271 | Potency | 1.049 | uM | ALA3562067 | active | nM | ||||
8. | PF-562271 | PF-562271 | Potency | 3.347 | uM | ALA3214813 | inactive | nM | ||||
9. | PF-562271 | PF-562271 | IC50 | = | 1.5 | nM | ALA4021282 | 8.82 | nM | Homo sapiens | ||
10. | PF-562271 | PF-562271 | IC50 | = | 13 | nM | ALA4021283 | 7.89 | nM | Homo sapiens | ||
11. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991926 | Inactive | nM | Homo sapiens | ||
12. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991925 | Inactive | nM | Homo sapiens | ||
13. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
14. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991923 | Inactive | nM | Homo sapiens | ||
15. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991922 | Inactive | nM | Homo sapiens | ||
16. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991921 | Inactive | nM | Homo sapiens | ||
17. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991920 | Inactive | nM | Homo sapiens | ||
18. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991919 | Inactive | nM | Homo sapiens | ||
19. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991917 | Inactive | nM | Homo sapiens | ||
20. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991916 | Inactive | nM | Homo sapiens |