# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1086077 | 46 | Intrinsic activity | = | 1.1 | % | ALA1117709 | % | Homo sapiens | |||
2. | ALA1086077 | 46 | EC50 | = | 385 | nM | ALA1117708 | 6.42 | nM | Homo sapiens | ||
3. | ALA1086077 | 46 | IC50 | = | 32 | nM | ALA1117707 | 7.50 | nM | Homo sapiens | ||
4. | ALA1086077 | 46 | Intrinsic activity | = | 0.2 | % | ALA1120621 | % | Homo sapiens | |||
5. | ALA1086077 | 46 | EC50 | = | 310 | nM | ALA1120620 | 6.51 | nM | Homo sapiens | ||
6. | ALA1086077 | 46 | t1/2 | = | 7.5 | hr | ALA1117717 | hr | Rattus norvegicus | |||
7. | ALA1086077 | 46 | Cmax | = | 290 | nM | ALA1117716 | nM | Rattus norvegicus | |||
8. | ALA1086077 | 46 | ED50 | = | 19 | uM | ALA1117715 | uM | Homo sapiens | |||
9. | ALA1086077 | 46 | ED50 | = | 9 | uM | ALA1117714 | uM | Homo sapiens | |||
10. | ALA1086077 | 46 | Activity | 0 | ALA1117713 | Active | ||||||
11. | ALA1086077 | 46 | solubility | = | 10 | uM | ALA1117712 | nM | ||||
12. | ALA1086077 | 46 | solubility | = | 180 | uM | ALA1117711 | nM | ||||
13. | ALA1086077 | 46 | Ki | = | 250 | nM | ALA1120619 | 6.60 | nM | Homo sapiens | ||
14. | ALA1086077 | 46 | Ki | = | 0.3 | nM | ALA1120618 | 9.52 | nM | Homo sapiens | ||
15. | ALA1086077 | 46 | Ki | = | 32 | nM | ALA1120617 | 7.50 | nM | Homo sapiens |