# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | XAV-939 | 1, XAV939 | IC50 | = | 114 | nM | ALA5227340 | 6.94 | nM | Homo sapiens | ||
2. | XAV-939 | 1, XAV939 | IC50 | = | 2.194 | nM | ALA5227339 | 8.66 | nM | Homo sapiens | ||
3. | XAV-939 | 1, XAV939 | IC50 | = | 4 | nM | ALA5227338 | 8.40 | nM | Homo sapiens | ||
4. | XAV-939 | 1, XAV939 | IC50 | = | 11 | nM | ALA5227337 | 7.96 | nM | Homo sapiens | ||
5. | XAV-939 | 1, XAV939 | Kd | = | 1.2 | uM | ALA5227336 | 5.92 | nM | Homo sapiens | ||
6. | XAV-939 | 1, XAV939 | Ki | = | 100 | nM | ALA5227335 | 7.00 | nM | Homo sapiens | ||
7. | XAV-939 | 1, XAV939 | Ki | = | 100 | nM | ALA5227334 | 7.00 | nM | Homo sapiens | ||
8. | XAV-939 | 1, XAV939 | INH | 0 | ALA5123654 | Active | % | |||||
9. | XAV-939 | 1, XAV939 | INH | 0 | ALA5123653 | Active | % | |||||
10. | XAV-939 | 1, XAV939 | INH | 0 | ALA5123650 | Active | % | |||||
11. | XAV-939 | 1, XAV939 | IC50 | = | 2.1 | nM | ALA5123649 | 8.68 | nM | Homo sapiens | ||
12. | XAV-939 | 1, XAV939 | IC50 | = | 1.9 | nM | ALA5123648 | 8.72 | nM | Homo sapiens | ||
13. | XAV-939 | 1, XAV939 | INH | = | 85 | % | ALA5123646 | % | Homo sapiens | |||
14. | XAV-939 | 1, XAV939 | INH | = | 86 | % | ALA5123645 | % | Homo sapiens | |||
15. | XAV-939 | 1, XAV939 | IC50 | = | 0.114 | uM | ALA5122239 | 6.94 | nM | Homo sapiens | ||
16. | XAV-939 | 1, XAV939 | IC50 | = | 2.194 | uM | ALA5122238 | nM | Homo sapiens | |||
17. | XAV-939 | 1, XAV939 | IC50 | = | 0.004 | uM | ALA5122237 | 8.40 | nM | Homo sapiens | ||
18. | XAV-939 | 1, XAV939 | IC50 | = | 0.011 | uM | ALA5122236 | 7.96 | nM | Homo sapiens | ||
19. | XAV-939 | 1, XAV939 | INH | = | 100 | % | ALA3382568 | % | Homo sapiens | |||
20. | XAV-939 | 1, XAV939 | INH | = | 91 | % | ALA3382567 | % | Homo sapiens |