# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | MF-766 | 9a, MF766 | Ratio Ki | > | 7000 | ALA1117801 | ||||||
2. | MF-766 | 9a, MF766 | Ratio Ki | > | 7000 | ALA1117800 | ||||||
3. | MF-766 | 9a, MF766 | Ratio Ki | > | 7000 | ALA1117799 | ||||||
4. | MF-766 | 9a, MF766 | Ratio Ki | > | 7000 | ALA1117798 | ||||||
5. | MF-766 | 9a, MF766 | Ratio Ki | > | 7000 | ALA1117797 | ||||||
6. | MF-766 | 9a, MF766 | Ratio Ki | > | 7000 | ALA1117796 | ||||||
7. | MF-766 | 9a, MF766 | Ratio Ki | > | 7000 | ALA1117795 | ||||||
8. | MF-766 | 9a, MF766 | Ratio Ki | > | 7000 | ALA1117794 | ||||||
9. | MF-766 | 9a, MF766 | Activity | = | 100 | % | ALA1117793 | % | Rattus norvegicus | |||
10. | MF-766 | 9a, MF766 | Activity | = | 70 | % | ALA1117792 | % | Rattus norvegicus | |||
11. | MF-766 | 9a, MF766 | Drug uptake | = | 3.1 | nM | ALA1117791 | nM | Rattus norvegicus | |||
12. | MF-766 | 9a, MF766 | Drug uptake | = | 28 | nM | ALA1117790 | nM | Rattus norvegicus | |||
13. | MF-766 | 9a, MF766 | ED100 | = | 0.025 | mg/kg/day | ALA1117789 | mg/kg/day | Rattus norvegicus | |||
14. | MF-766 | 9a, MF766 | ED100 | = | 0.025 | mg/kg/day | ALA1117788 | mg/kg/day | Rattus norvegicus | |||
15. | MF-766 | 9a, MF766 | ED50 | = | 0.004 | mg/kg/day | ALA1117787 | mg/kg/day | Rattus norvegicus | |||
16. | MF-766 | 9a, MF766 | Activity | = | 50 | pmolequiv/mg | ALA1117786 | pmolequiv/mg | Homo sapiens | |||
17. | MF-766 | 9a, MF766 | Activity | = | 61 | pmolequiv/mg | ALA1117785 | pmolequiv/mg | Rattus norvegicus | |||
18. | MF-766 | 9a, MF766 | AUC | = | 15 | uM.hr | ALA1117784 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Canis lupus familiaris | ||
19. | MF-766 | 9a, MF766 | AUC | = | 150 | uM.hr | ALA1117783 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
20. | MF-766 | 9a, MF766 | F | = | 74 | % | ALA1117782 | % | Canis lupus familiaris |