| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA296435 | (+)-2S,3R EHNA | Ki | = | 1 | nM | ALA5152123 | 9.00 | nM | Homo sapiens | ||
| 2. | ALA296435 | (+)-2S,3R EHNA | IC50 | = | 800 | nM | ALA4373106 | 6.10 | nM | Homo sapiens | ||
| 3. | ALA296435 | (+)-2S,3R EHNA | IC50 | = | 2.62 | uM | ALA4733110 | 5.58 | nM | Homo sapiens | ||
| 4. | ALA296435 | (+)-2S,3R EHNA | IC50 | = | 2.46 | uM | ALA4182273 | 5.61 | nM | Homo sapiens | ||
| 5. | ALA296435 | (+)-2S,3R EHNA | IC50 | = | 800 | nM | ALA4182275 | 6.10 | nM | |||
| 6. | ALA296435 | (+)-2S,3R EHNA | INH | = | 37.45 | % | ALA4182274 | % | Homo sapiens | |||
| 7. | ALA296435 | (+)-2S,3R EHNA | CL | 0 | ALA4179248 | Bld | Rattus norvegicus | |||||
| 8. | ALA296435 | (+)-2S,3R EHNA | Cp | 0 | ALA4179247 | Bld | Rattus norvegicus | |||||
| 9. | ALA296435 | (+)-2S,3R EHNA | AUCt | = | 0.35 | uM.hr | ALA4179239 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 10. | ALA296435 | (+)-2S,3R EHNA | Ki | = | 2.2 | nM | ALA4179226 | 8.66 | nM | Bos taurus | ||
| 11. | ALA296435 | (+)-2S,3R EHNA | IC50 | = | 0.8 | uM | ALA3772722 | 6.10 | nM | Homo sapiens | ||
| 12. | ALA296435 | (+)-2S,3R EHNA | IC50 | = | 2 | uM | ALA3772723 | 5.70 | nM | |||
| 13. | ALA296435 | (+)-2S,3R EHNA | IC50 | = | 0.7 | uM | ALA3772724 | 6.16 | nM | |||
| 14. | ALA296435 | (+)-2S,3R EHNA | IC50 | = | 1.7 | uM | ALA3772725 | 5.77 | nM | Homo sapiens | ||
| 15. | ALA296435 | (+)-2S,3R EHNA | Ki | = | 1.14 | nM | ALA1013499 | 8.94 | nM | |||
| 16. | ALA296435 | (+)-2S,3R EHNA | Solubility | > | 65 | ug ml-1 | ALA860265 | ug.mL-1 | Homo sapiens | |||
| 17. | ALA296435 | (+)-2S,3R EHNA | Papp | 0 | ALA860263 | Not Determined | Canis lupus familiaris | |||||
| 18. | ALA296435 | (+)-2S,3R EHNA | Papp | 0 | ALA860262 | Not Determined | Canis lupus familiaris | |||||
| 19. | ALA296435 | (+)-2S,3R EHNA | Papp | = | 18 | ucm/s | ALA860260 | ucm/s | Homo sapiens | |||
| 20. | ALA296435 | (+)-2S,3R EHNA | Papp | = | 34 | ucm/s | ALA860259 | ucm/s | Homo sapiens |
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