# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1159715 | 1, (+/-)-Th 1206 | pIC50 | < | 4.7 | ALA4651403 | No. Measurements = 1 | nM | Severe acute respiratory syndrome coronavirus 2 | |||
2. | ALA1159715 | 1, (+/-)-Th 1206 | IC50 | > | 0 | M | ALA4651403 | No. Measurements = 1 | nM | Severe acute respiratory syndrome coronavirus 2 | ||
3. | ALA1159715 | 1, (+/-)-Th 1206 | Ratio | = | 53 | ALA5119563 | Homo sapiens | |||||
4. | ALA1159715 | 1, (+/-)-Th 1206 | Intrinsic activity | = | 1 | ALA3280907 | Cavia porcellus | |||||
5. | ALA1159715 | 1, (+/-)-Th 1206 | Selectivity ratio | = | 5.5 | ALA3280906 | ||||||
6. | ALA1159715 | 1, (+/-)-Th 1206 | Intrinsic activity | = | 1 | ALA3280905 | Cavia porcellus | |||||
7. | ALA1159715 | 1, (+/-)-Th 1206 | ED50 | = | 1.3 | nM | ALA3280902 | 8.89 | nM | Cavia porcellus | ||
8. | ALA1159715 | 1, (+/-)-Th 1206 | ED25 | = | 7.1 | nM | ALA3280903 | nM | Cavia porcellus | |||
9. | ALA1159715 | 1, (+/-)-Th 1206 | Ratio | = | 5.5 | ALA3283663 | ||||||
10. | ALA1159715 | 1, (+/-)-Th 1206 | Ratio | = | 1 | ALA3283662 | ||||||
11. | ALA1159715 | 1, (+/-)-Th 1206 | Ratio | = | 1 | ALA3283661 | ||||||
12. | ALA1159715 | 1, (+/-)-Th 1206 | ED25 | = | 7.1 | nM | ALA3283655 | nM | ||||
13. | ALA1159715 | 1, (+/-)-Th 1206 | ED50 | = | 1.3 | nM | ALA3283652 | 8.89 | nM | |||
14. | ALA1159715 | 1, (+/-)-Th 1206 | clogP | = | 1.03 | ALA856958 | ||||||
15. | ALA1159715 | 1, (+/-)-Th 1206 | Log 1/ISA | = | 0.17 | ALA885386 | ||||||
16. | ALA1159715 | 1, (+/-)-Th 1206 | ISA | = | 0.68 | ALA653454 | Bos taurus | |||||
17. | ALA1159715 | 1, (+/-)-Th 1206 | cAMP production | = | 83 | pM min-1 mg-1 | ALA655183 | pM min-1 mg-1 | Bos taurus | |||
18. | ALA1159715 | 1, (+/-)-Th 1206 | Concentration | = | 3 | M | ALA651195 | M | Bos taurus | |||
19. | ALA1159715 | 1, (+/-)-Th 1206 | KD app | = | 0.67 | uM | ALA651194 | uM | Bos taurus | |||
20. | ALA1159715 | 1, (+/-)-Th 1206 | -Delta G | = | 9.29 | ALA819725 | Bos taurus |