Activities

#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Comment	Assay	Assay Organism
1.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		29.093	uM	ALA2354282		inactive	nM	Homo sapiens
2.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		35.481	uM	ALA2114784		inconclusive	nM	Homo sapiens
3.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	IC50	=	0.25	uM	ALA3389217	6.60		nM	Homo sapiens
4.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		26.855	uM	ALA3215185		active	nM	Homo sapiens
5.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		2.502	uM	ALA3215169		inconclusive	nM
6.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		39.811	uM	ALA3214909		inconclusive	nM
7.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		3.965	uM	ALA3214913		inconclusive	nM
8.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		28.184	uM	ALA3214837		inconclusive	nM
9.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		0.947	uM	ALA1613922		Active	nM	Homo sapiens
10.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		29.081	uM	ALA1738675		inconclusive	nM	Homo sapiens
11.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		2.393	uM	ALA1738600		Active	nM	Homo sapiens
12.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		18.356	uM	ALA1614015		inconclusive	nM
13.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		5.358	uM	ALA1738509		Active	nM	Trypanosoma brucei brucei
14.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		1.259	uM	ALA1738610		Active	nM	Homo sapiens
15.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		2.393	uM	ALA1614279		Active	nM	Trypanosoma brucei
16.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		1	uM	ALA1738442		Active	nM	Homo sapiens
17.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		5.323	uM	ALA1614194		Active	nM	Bacillus subtilis (strain 168)
18.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		100	uM	ALA1614315		inconclusive	nM	Homo sapiens
19.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		29.935	uM	ALA1794424		inconclusive	nM	Rattus norvegicus
20.	1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid	Cibacron blue(para)	Potency		28.184	uM	ALA1794367		inconclusive	nM	Homo sapiens

1.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

29.093

uM

ALA2354282

inactive

nM

Homo sapiens

2.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

35.481

uM

ALA2114784

inconclusive

nM

Homo sapiens

3.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

IC50

=

0.25

uM

ALA3389217

6.60

nM

Homo sapiens

4.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

26.855

uM

ALA3215185

active

nM

Homo sapiens

5.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

2.502

uM

ALA3215169

inconclusive

nM

6.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

39.811

uM

ALA3214909

inconclusive

nM

7.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

3.965

uM

ALA3214913

inconclusive

nM

8.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

28.184

uM

ALA3214837

inconclusive

nM

9.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

0.947

uM

ALA1613922

Active

nM

Homo sapiens

10.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

29.081

uM

ALA1738675

inconclusive

nM

Homo sapiens

11.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

2.393

uM

ALA1738600

Active

nM

Homo sapiens

12.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

18.356

uM

ALA1614015

inconclusive

nM

13.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

5.358

uM

ALA1738509

Active

nM

Trypanosoma brucei brucei

14.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

1.259

uM

ALA1738610

Active

nM

Homo sapiens

15.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

2.393

uM

ALA1614279

Active

nM

Trypanosoma brucei

16.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

1

uM

ALA1738442

Active

nM

Homo sapiens

17.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

5.323

uM

ALA1614194

Active

nM

Bacillus subtilis (strain 168)

18.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

100

uM

ALA1614315

inconclusive

nM

Homo sapiens

19.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

29.935

uM

ALA1794424

inconclusive

nM

Rattus norvegicus

20.

1-Amino-4-((4-((4-chloro-6-((4-sulfophenyl)amino)-1,3,5-triazin-2-yl)amino)-3-sulfophenyl)amino)-9,10-dihydro-9,10-dioxo-2-anthracenesulfonic acid

Cibacron blue(para)

Potency

28.184

uM

ALA1794367

inconclusive

nM

Homo sapiens