# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA42205 | 80 (ICA-15451) | Activity | = | 47 | % | ALA948126 | % | Mus musculus | |||
2. | ALA42205 | 80 (ICA-15451) | Activity | = | 44.5 | % | ALA948125 | % | Mus musculus | |||
3. | ALA42205 | 80 (ICA-15451) | Activity | = | 27 | g/dl | ALA948124 | g/dl | Mus musculus | |||
4. | ALA42205 | 80 (ICA-15451) | Activity | = | 34 | g/dl | ALA948123 | g/dl | Mus musculus | |||
5. | ALA42205 | 80 (ICA-15451) | Activity | = | 2 | mmol | ALA948122 | mmol | Mus musculus | |||
6. | ALA42205 | 80 (ICA-15451) | Activity | = | 4 | mmol | ALA948121 | mmol | Mus musculus | |||
7. | ALA42205 | 80 (ICA-15451) | IC50 | = | 9 | nM | ALA948111 | 8.05 | nM | Homo sapiens | ||
8. | ALA42205 | 80 (ICA-15451) | Inhibition | < | 20 | % | ALA948119 | % | Homo sapiens | |||
9. | ALA42205 | 80 (ICA-15451) | Cmax | = | 250 | ng/ml | ALA948117 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
10. | ALA42205 | 80 (ICA-15451) | Tmax | = | 2 | hr | ALA948116 | hr | Rattus norvegicus | |||
11. | ALA42205 | 80 (ICA-15451) | t1/2 | = | 2.5 | hr | ALA948115 | hr | Rattus norvegicus | |||
12. | ALA42205 | 80 (ICA-15451) | F | = | 35 | % | ALA948114 | % | Rattus norvegicus | |||
13. | ALA42205 | 80 (ICA-15451) | Solubility | = | 5.8 | uM | ALA948113 | nM | ||||
14. | ALA42205 | 80 (ICA-15451) | Compound remaining | = | 40 | % | ALA948112 | % | Rattus norvegicus | |||
15. | ALA42205 | 80 (ICA-15451) | IC50 | = | 2000 | nM | ALA819394 | 5.70 | nM | Homo sapiens | ||
16. | ALA42205 | 80 (ICA-15451) | IC50 | = | 9 | nM | ALA680747 | 8.05 | nM | Homo sapiens |