| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1201187 | 13, UK-427857 | beta t1/2 | = | 53.23 | hr | ALA5231706 | hr | ||||
| 2. | ALA1201187 | 13, UK-427857 | AUC | = | 567.17 | ng.hr/ml | ALA5231705 | ng.hr.mL-1 | ||||
| 3. | ALA1201187 | 13, UK-427857 | IC50 | = | 14.9 | uM | ALA5154066 | 4.83 | nM | Homo sapiens | ||
| 4. | ALA1201187 | 13, UK-427857 | IC50 | = | 3.1 | uM | ALA5154065 | 5.51 | nM | Homo sapiens | ||
| 5. | ALA1201187 | 13, UK-427857 | IC50 | > | 25 | uM | ALA5154064 | nM | Homo sapiens | |||
| 6. | ALA1201187 | 13, UK-427857 | IC50 | > | 25 | uM | ALA5154063 | nM | Homo sapiens | |||
| 7. | ALA1201187 | 13, UK-427857 | IC50 | = | 14.4 | uM | ALA5154062 | 4.84 | nM | Homo sapiens | ||
| 8. | ALA1201187 | 13, UK-427857 | IC50 | > | 25 | uM | ALA5154061 | nM | Homo sapiens | |||
| 9. | ALA1201187 | 13, UK-427857 | CL | = | 74 | ml/min/mg | ALA5154060 | mL.min-1.g-1 | ||||
| 10. | ALA1201187 | 13, UK-427857 | t1/2 | = | 0.9 | hr | ALA5154059 | hr | ||||
| 11. | ALA1201187 | 13, UK-427857 | t1/2 | = | 0.9 | hr | ALA5154054 | hr | ||||
| 12. | ALA1201187 | 13, UK-427857 | AUC | = | 12.4 | ng.hr/ml | ALA5154051 | ng.hr.mL-1 | ||||
| 13. | ALA1201187 | 13, UK-427857 | Tmax | = | 2 | hr | ALA5154048 | hr | ||||
| 14. | ALA1201187 | 13, UK-427857 | Cmax | = | 5.5 | ng/ml | ALA5154047 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 15. | ALA1201187 | 13, UK-427857 | EC50 | = | 2.18 | nM | ALA5154035 | 8.66 | nM | Human immunodeficiency virus 1 | ||
| 16. | ALA1201187 | 13, UK-427857 | TI | > | 2173.91 | ALA5154034 | ||||||
| 17. | ALA1201187 | 13, UK-427857 | EC50 | = | 92 | nM | ALA5154033 | 7.04 | nM | Human immunodeficiency virus 1 | ||
| 18. | ALA1201187 | 13, UK-427857 | TI | > | 13404.83 | ALA5154032 | ||||||
| 19. | ALA1201187 | 13, UK-427857 | EC50 | = | 14.92 | nM | ALA5154031 | 7.83 | nM | Human immunodeficiency virus 1 | ||
| 20. | ALA1201187 | 13, UK-427857 | TI | > | 19704.43 | ALA5154030 |
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