| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1207972 | 7 | Fu | = | 0.002 | % | ALA4702833 | |||||
| 2. | ALA1207972 | 7 | CLH | = | 2 | ml/min.kg | ALA4702832 | mL.min-1.kg-1 | ||||
| 3. | ALA1207972 | 7 | CLH | = | 19.5 | ml/min.kg | ALA4702831 | mL.min-1.kg-1 | ||||
| 4. | ALA1207972 | 7 | Ratio | = | 0.654 | ALA4702829 | ||||||
| 5. | ALA1207972 | 7 | Ratio | = | 0.561 | ALA4702828 | ||||||
| 6. | ALA1207972 | 7 | Fu | = | 0.003 | % | ALA4702826 | |||||
| 7. | ALA1207972 | 7 | CLH | = | 180 | ml/min.kg | ALA4702824 | mL.min-1.kg-1 | ||||
| 8. | ALA1207972 | 7 | logD | = | 2.1 | ALA4702823 | ||||||
| 9. | ALA1207972 | 7 | Papp | = | 12 | 10^-6 cm/s | ALA4702822 | 10^-6 cm/s | ||||
| 10. | ALA1207972 | 7 | pKa | = | 5.3 | ALA4702821 | ||||||
| 11. | ALA1207972 | 7 | Kd | = | 47.9 | nM | ALA2320404 | 7.32 | nM | Mus musculus | ||
| 12. | ALA1207972 | 7 | pKi | = | 5.76 | ALA2320402 | 5.76 | nM | Mus musculus | |||
| 13. | ALA1207972 | 7 | pKi | < | 6 | ALA2320403 | nM | Mus musculus | ||||
| 14. | ALA1207972 | 7 | pKi | < | 6 | ALA2320401 | nM | Mus musculus | ||||
| 15. | ALA1207972 | 7 | pKi | < | 6 | ALA2320400 | nM | Mus musculus | ||||
| 16. | ALA1207972 | 7 | Ratio IC50 | = | 100 | ALA2320405 | ||||||
| 17. | ALA1207972 | 7 | t1/2 | = | 65 | min | ALA2320398 | hr | Mus musculus | |||
| 18. | ALA1207972 | 7 | CL | = | 59.2 | ml/min.Kg | ALA2320399 | mL.min-1.kg-1 | Mus musculus | |||
| 19. | ALA1207972 | 7 | Vdss | = | 0.9 | L/Kg | ALA2320397 | L.kg-1 | Mus musculus | |||
| 20. | ALA1207972 | 7 | F | = | 13.8 | % | ALA2320395 | % | Mus musculus |
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