| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1224147 | R3C2 Table 5 | EC50 | = | 1.6 | uM | ALA1228892 | 5.80 | nM | Rattus norvegicus | ||
| 2. | ALA1224147 | R3C2 Table 5 | t1/2 | = | 0.05 | hr | ALA1228891 | hr | Rattus norvegicus | |||
| 3. | ALA1224147 | R3C2 Table 5 | Vd | = | 0.07 | L/Kg | ALA1228890 | L.kg-1 | Rattus norvegicus | |||
| 4. | ALA1224147 | R3C2 Table 5 | Cmax | = | 9700 | ng/ml | ALA1228889 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 5. | ALA1224147 | R3C2 Table 5 | CL | = | 30 | ml/min.kg | ALA1225931 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 6. | ALA1224147 | R3C2 Table 5 | CL | = | 18 | microL/min/mg | ALA1225930 | mL.min-1.g-1 | Rattus norvegicus | |||
| 7. | ALA1224147 | R3C2 Table 5 | CL | = | 11 | microL/min/mg | ALA1225929 | mL.min-1.g-1 | Homo sapiens | |||
| 8. | ALA1224147 | R3C2 Table 5 | IC50 | = | 2.7 | uM | ALA1225928 | 5.57 | nM | Rattus norvegicus | ||
| 9. | ALA1224147 | R3C2 Table 5 | EC50 | = | 2.5 | uM | ALA1225927 | 5.60 | nM | Homo sapiens | ||
| 10. | ALA1224147 | R3C2 Table 5 | IC50 | > | 50 | uM | ALA1225926 | nM | Homo sapiens | |||
| 11. | ALA1224147 | R3C2 Table 5 | IC50 | = | 0.63 | uM | ALA1225925 | 6.20 | nM | Homo sapiens |
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