| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Activity | 0 | ALA4150362 | Active | Cricetulus griseus | |||||
| 2. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Activity | 0 | ALA4150365 | Active | Cricetulus griseus | |||||
| 3. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Activity | 0 | ALA4150364 | Active | Cricetulus griseus | |||||
| 4. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Activity | 0 | ALA4150363 | Active | Cricetulus griseus | |||||
| 5. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Activity | 0 | ALA4150361 | Active | Cricetulus griseus | |||||
| 6. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Ki | = | 49 | uM | ALA2184190 | 4.31 | nM | |||
| 7. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | IC50 | = | 80 | uM | ALA962639 | 4.10 | nM | Homo sapiens | ||
| 8. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | IC50 | = | 40 | uM | ALA962638 | 4.40 | nM | Homo sapiens | ||
| 9. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | IC50 | 0 | ALA970838 | Not Determined | Homo sapiens | |||||
| 10. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | IC50 | = | 38.4 | ug ml-1 | ALA970837 | ug.mL-1 | Rattus norvegicus | |||
| 11. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Activity | 0 | ALA948574 | Not Active | Mus musculus | |||||
| 12. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | IC50 | = | 23.5 | uM | ALA948572 | 4.63 | nM | Mus musculus | ||
| 13. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | IC50 | = | 5.4 | uM | ALA923068 | 5.27 | nM | Plasmodium falciparum | ||
| 14. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | IC50 | > | 69 | uM | ALA923067 | nM | Plasmodium falciparum | |||
| 15. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | IC50 | > | 500 | uM | ALA923066 | nM | Plasmodium falciparum | |||
| 16. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Activity | = | 7 | % | ALA1062022 | Antagonist | % | Homo sapiens | ||
| 17. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Activity | = | 96 | % | ALA1063666 | % | Homo sapiens | |||
| 18. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Activity | = | 88 | % | ALA1061099 | % | Homo sapiens | |||
| 19. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Activity | = | 36 | % | ALA1061974 | Antagonist | % | Homo sapiens | ||
| 20. | ALA1233654 | H-7 (1-(5-isoquinolinesulfonyl)-2-methylpiperazine) | Activity | = | 80 | % | ALA1060207 | % | Homo sapiens |
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