| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1233845 | 1, GS-8374 | CLH | = | 1 | microL/min/mg | ALA3225593 | mL.min-1.g-1 | Homo sapiens | |||
| 2. | ALA1233845 | 1, GS-8374 | CLH | = | 2.6 | microL/min/mg | ALA3225592 | mL.min-1.g-1 | Homo sapiens | |||
| 3. | ALA1233845 | 1, GS-8374 | CLH | = | 9.2 | microL/min/mg | ALA3225590 | mL.min-1.g-1 | Homo sapiens | |||
| 4. | ALA1233845 | 1, GS-8374 | F | = | 100 | % | ALA3225589 | % | Canis lupus familiaris | |||
| 5. | ALA1233845 | 1, GS-8374 | F | = | 6.9 | % | ALA3225588 | % | Canis lupus familiaris | |||
| 6. | ALA1233845 | 1, GS-8374 | CL | = | 2.13 | L/hr/kg | ALA3225587 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 7. | ALA1233845 | 1, GS-8374 | Ratio EC50 | = | 0.6 | ALA3225586 | Human immunodeficiency virus 1 | |||||
| 8. | ALA1233845 | 1, GS-8374 | Ratio EC50 | = | 0.2 | ALA3225585 | Human immunodeficiency virus 1 | |||||
| 9. | ALA1233845 | 1, GS-8374 | Ratio EC50 | = | 0.9 | ALA3225584 | Human immunodeficiency virus 1 | |||||
| 10. | ALA1233845 | 1, GS-8374 | Ratio EC50 | = | 0.1 | ALA3225583 | Human immunodeficiency virus 1 | |||||
| 11. | ALA1233845 | 1, GS-8374 | FC | = | 15 | ALA3225578 | Human immunodeficiency virus 1 | |||||
| 12. | ALA1233845 | 1, GS-8374 | CC50 | = | 61.3 | uM | ALA3225582 | nM | Homo sapiens | |||
| 13. | ALA1233845 | 1, GS-8374 | CC50 | > | 100 | uM | ALA3225581 | nM | Homo sapiens | |||
| 14. | ALA1233845 | 1, GS-8374 | Ratio EC50 | = | 2.4 | ALA3225580 | Human immunodeficiency virus 1 | |||||
| 15. | ALA1233845 | 1, GS-8374 | Ratio EC50 | = | 0.7 | ALA3225577 | Human immunodeficiency virus 1 | |||||
| 16. | ALA1233845 | 1, GS-8374 | Ratio EC50 | = | 2.7 | ALA3225579 | Human immunodeficiency virus 1 | |||||
| 17. | ALA1233845 | 1, GS-8374 | EC50 | = | 3.5 | nM | ALA3227406 | 8.46 | nM | Human immunodeficiency virus 1 | ||
| 18. | ALA1233845 | 1, GS-8374 | Ki | = | 8.1 | pM | ALA3227405 | nM | Human immunodeficiency virus 1 | |||
| 19. | ALA1233845 | 1, GS-8374 | Ki | = | 170 | nM | ALA5036786 | 6.77 | nM | |||
| 20. | ALA1233845 | 1, GS-8374 | EC50 | = | 3.5 | nM | ALA5252992 | 8.46 | nM | Human immunodeficiency virus 1 |
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