# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1235128 | 1d | Selectivity Index | = | 1.9 | ALA4689560 | ||||||
2. | ALA1235128 | 1d | Ki | = | 1.8 | uM | ALA4689557 | 5.75 | nM | Homo sapiens | ||
3. | ALA1235128 | 1d | Kd | = | 29 | uM | ALA4689557 | 4.54 | nM | Homo sapiens | ||
4. | ALA1235128 | 1d | Ki | = | 3.2 | uM | ALA4689556 | 5.50 | nM | Homo sapiens | ||
5. | ALA1235128 | 1d | Kd | = | 16 | uM | ALA4689556 | 4.80 | nM | Homo sapiens | ||
6. | ALA1235128 | 1d | pKi | = | 7.3 | ALA3790454 | 7.30 | nM | Homo sapiens | |||
7. | ALA1235128 | 1d | Ratio Ki | = | 17.5 | ALA2072281 | ||||||
8. | ALA1235128 | 1d | Efficacy | = | 78.6 | % | ALA2072282 | % | Homo sapiens | |||
9. | ALA1235128 | 1d | Ki | = | 550 | nM | ALA2072278 | 6.26 | nM | Rattus norvegicus | ||
10. | ALA1235128 | 1d | Ki | = | 1240 | nM | ALA2072277 | 5.91 | nM | Rattus norvegicus | ||
11. | ALA1235128 | 1d | Ki | = | 50 | nM | ALA2072276 | 7.30 | nM | Homo sapiens | ||
12. | ALA1235128 | 1d | Ki | = | 210 | nM | ALA2072275 | 6.68 | nM | Homo sapiens | ||
13. | ALA1235128 | 1d | Ki | = | 12 | nM | ALA2072274 | 7.92 | nM | Homo sapiens | ||
14. | ALA1235128 | 1d | EC50 | = | 29 | uM | ALA639461 | 4.54 | nM | Homo sapiens | ||
15. | ALA1235128 | 1d | Ki | = | 44 | nM | ALA646602 | 7.36 | nM | Homo sapiens | ||
16. | ALA1235128 | 1d | Ki | = | 550 | nM | ALA641310 | 6.26 | nM | Rattus norvegicus | ||
17. | ALA1235128 | 1d | GTP shift | = | 3.2 | ALA842883 | ||||||
18. | ALA1235128 | 1d | Ki | = | 3960 | nM | ALA640468 | 5.40 | nM | Rattus norvegicus | ||
19. | ALA1235128 | 1d | Ki | = | 1240 | nM | ALA640467 | 5.91 | nM | Rattus norvegicus | ||
20. | ALA1235128 | 1d | Ki | = | 31 | nM | ALA754752 | 7.51 | nM | Rattus norvegicus |