# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1236475 | 5, THU, Epimeric mixture | Inhibition | = | 45.2 | % | ALA4303805 | % | Severe acute respiratory syndrome coronavirus 2 | |||
2. | ALA1236475 | 5, THU, Epimeric mixture | inhibition | = | -0.09 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
3. | ALA1236475 | 5, THU, Epimeric mixture | Drug degradation | = | 80 | % | ALA3242114 | % | ||||
4. | ALA1236475 | 5, THU, Epimeric mixture | Drug degradation | = | 50 | % | ALA3242113 | % | ||||
5. | ALA1236475 | 5, THU, Epimeric mixture | Stability | = | 15 | % | ALA3242112 | % | ||||
6. | ALA1236475 | 5, THU, Epimeric mixture | Stability | = | 50 | % | ALA3241964 | % | ||||
7. | ALA1236475 | 5, THU, Epimeric mixture | Ki | = | 440 | uM | ALA3241963 | nM | Homo sapiens | |||
8. | ALA1236475 | 5, THU, Epimeric mixture | IC50 | = | 0.34 | uM | ALA3241962 | 6.47 | nM | Homo sapiens | ||
9. | ALA1236475 | 5, THU, Epimeric mixture | inhibition | = | -0.09 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
10. | ALA1236475 | 5, THU, Epimeric mixture | Inhibition | = | 13.165 | % | ALA4495582 | % | Severe acute respiratory syndrome coronavirus 2 |