| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1237000 | 5, MK-0536 | CL | = | 2.2 | ml/min.kg | ALA5237343 | mL.min-1.kg-1 | ||||
| 2. | ALA1237000 | 5, MK-0536 | CL | = | 2.3 | ml/min.kg | ALA5237342 | mL.min-1.kg-1 | ||||
| 3. | ALA1237000 | 5, MK-0536 | EC50 | = | 1 | nM | ALA5237341 | 9.00 | nM | Human immunodeficiency virus | ||
| 4. | ALA1237000 | 5, MK-0536 | EC50 | = | 2 | nM | ALA5237340 | 8.70 | nM | Human immunodeficiency virus | ||
| 5. | ALA1237000 | 5, MK-0536 | FC | = | 1 | ALA5237339 | Human immunodeficiency virus | |||||
| 6. | ALA1237000 | 5, MK-0536 | EC50 | = | 3 | nM | ALA5237338 | 8.52 | nM | Human immunodeficiency virus | ||
| 7. | ALA1237000 | 5, MK-0536 | EC50 | = | 1 | nM | ALA5237336 | 9.00 | nM | Human immunodeficiency virus | ||
| 8. | ALA1237000 | 5, MK-0536 | CLH | < | 20 | ml/min.kg | ALA3625845 | mL.min-1.kg-1 | Homo sapiens | |||
| 9. | ALA1237000 | 5, MK-0536 | F | = | 44 | % | ALA3625844 | % | Canis lupus familiaris | |||
| 10. | ALA1237000 | 5, MK-0536 | CL | = | 2.2 | ml/min.kg | ALA3625166 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 11. | ALA1237000 | 5, MK-0536 | F | = | 29 | % | ALA3625165 | % | Rattus norvegicus | |||
| 12. | ALA1237000 | 5, MK-0536 | CL | = | 2.3 | ml/min.kg | ALA3625164 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 13. | ALA1237000 | 5, MK-0536 | Ratio IC50 | = | 3 | ALA3625163 | Human immunodeficiency virus 1 | |||||
| 14. | ALA1237000 | 5, MK-0536 | Ratio IC50 | = | 1 | ALA3625162 | Human immunodeficiency virus 1 | |||||
| 15. | ALA1237000 | 5, MK-0536 | Ratio IC50 | = | 1 | ALA3625161 | Human immunodeficiency virus 1 | |||||
| 16. | ALA1237000 | 5, MK-0536 | Ratio IC50 | = | 2 | ALA3625160 | Human immunodeficiency virus 1 | |||||
| 17. | ALA1237000 | 5, MK-0536 | Ratio IC50 | = | 1 | ALA3625159 | Human immunodeficiency virus 1 | |||||
| 18. | ALA1237000 | 5, MK-0536 | IP | = | 53 | nM | ALA3625042 | nM | Human immunodeficiency virus 1 | |||
| 19. | ALA1237000 | 5, MK-0536 | IP | = | 6 | nM | ALA3625041 | nM | Human immunodeficiency virus 1 |
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