# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | MEL57A | (R)-6 | Selectivity ratio | = | 30 | ALA1825381 | ||||||
2. | MEL57A | (R)-6 | Selectivity ratio | > | 150 | ALA1825380 | ||||||
3. | MEL57A | (R)-6 | EC50 | = | 113.2 | uM | ALA1250988 | nM | ||||
4. | MEL57A | (R)-6 | EC50 | = | 103.78 | uM | ALA1250987 | nM | Homo sapiens | |||
5. | MEL57A | (R)-6 | Selectivity ratio | = | 130 | ALA1250992 | ||||||
6. | MEL57A | (R)-6 | Selectivity ratio | = | 170 | ALA1250991 | ||||||
7. | MEL57A | (R)-6 | INH | = | 27 | % | ALA1250983 | % | Mus musculus | |||
8. | MEL57A | (R)-6 | INH | = | 93 | % | ALA1250985 | % | Homo sapiens | |||
9. | MEL57A | (R)-6 | EC50 | = | 0.6 | uM | ALA1250984 | 6.22 | nM | Mus musculus | ||
10. | MEL57A | (R)-6 | EC50 | = | 18.3 | uM | ALA1250986 | 4.74 | nM | Mus musculus |