# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1253992 | (R)-5 | EC50 | = | 7.1 | uM | ALA1250988 | 5.15 | nM | |||
2. | ALA1253992 | (R)-5 | EC50 | = | 24.94 | uM | ALA1250987 | 4.60 | nM | Homo sapiens | ||
3. | ALA1253992 | (R)-5 | Selectivity ratio | = | 10 | ALA1250990 | ||||||
4. | ALA1253992 | (R)-5 | Selectivity ratio | = | 4 | ALA1250989 | ||||||
5. | ALA1253992 | (R)-5 | EC50 | = | 2.3 | uM | ALA1250986 | 5.64 | nM | Mus musculus | ||
6. | ALA1253992 | (R)-5 | INH | = | 63 | % | ALA1250983 | % | Mus musculus | |||
7. | ALA1253992 | (R)-5 | INH | = | 83 | % | ALA1250985 | % | Homo sapiens | |||
8. | ALA1253992 | (R)-5 | EC50 | = | 9.41 | uM | ALA1250984 | 5.03 | nM | Mus musculus |