| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1254771 | 24 | PPB | 74.25 | % | ALA3301366 | % | |||||
| 2. | ALA1254771 | 24 | Vd | = | 1.4 | L/Kg | ALA2092284 | L.kg-1 | Rattus norvegicus | |||
| 3. | ALA1254771 | 24 | Vd | = | 2.6 | L/Kg | ALA2092283 | L.kg-1 | Mus musculus | |||
| 4. | ALA1254771 | 24 | CL | = | 27.4 | ml/min.kg | ALA2092281 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 5. | ALA1254771 | 24 | CL | = | 131 | ml/min.kg | ALA2092280 | mL.min-1.kg-1 | Mus musculus | |||
| 6. | ALA1254771 | 24 | pKb | = | 9.7 | ALA2092266 | Homo sapiens | |||||
| 7. | ALA1254771 | 24 | pKb | = | 8.2 | ALA2092267 | Mus musculus | |||||
| 8. | ALA1254771 | 24 | pKb | = | 9.5 | ALA2092268 | Oryctolagus cuniculus | |||||
| 9. | ALA1254771 | 24 | pKb | = | 8.1 | ALA2092269 | Rattus norvegicus | |||||
| 10. | ALA1254771 | 24 | Stability | = | 57 | % | ALA2092270 | % | ||||
| 11. | ALA1254771 | 24 | Papp | = | 1.3 | ucm/s | ALA2092273 | ucm/s | Homo sapiens | |||
| 12. | ALA1254771 | 24 | F | = | 12 | % | ALA2092274 | % | Mus musculus | |||
| 13. | ALA1254771 | 24 | t1/2 | = | 0.6 | hr | ALA2092277 | hr | Mus musculus | |||
| 14. | ALA1254771 | 24 | t1/2 | = | 2.1 | hr | ALA2092278 | hr | Rattus norvegicus | |||
| 15. | ALA1254771 | 24 | Ki | = | 0.3 | nM | ALA2092264 | 9.52 | nM | Homo sapiens | ||
| 16. | ALA1254771 | 24 | INH | = | 57 | % | ALA2091465 | % | Rattus norvegicus | |||
| 17. | ALA1254771 | 24 | INH | = | 52 | % | ALA2091467 | % | Rattus norvegicus | |||
| 18. | ALA1254771 | 24 | INH | = | 46 | % | ALA2091468 | % | Rattus norvegicus | |||
| 19. | ALA1254771 | 24 | Activity | = | 61 | % | ALA2091466 | % | Rattus norvegicus | |||
| 20. | ALA1254771 | 24 | Stability | = | 80 | % | ALA2091469 | % |
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