# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1258659 | 4-3 | IC50 | = | 2.18 | uM | ALA2380129 | 5.66 | nM | Homo sapiens | ||
2. | ALA1258659 | 4-3 | IC50 | = | 5.14 | uM | ALA2380128 | 5.29 | nM | Homo sapiens | ||
3. | ALA1258659 | 4-3 | IC50 | = | 6.31 | uM | ALA2380127 | 5.20 | nM | Homo sapiens | ||
4. | ALA1258659 | 4-3 | IC50 | = | 4.9 | uM | ALA2380126 | 5.31 | nM | Homo sapiens | ||
5. | ALA1258659 | 4-3 | IC50 | = | 5.26 | uM | ALA2380124 | 5.28 | nM | Homo sapiens | ||
6. | ALA1258659 | 4-3 | solubility | = | 1.1 | uM | ALA2380123 | nM | ||||
7. | ALA1258659 | 4-3 | permeability | 0 | ALA2380122 | Not Determined | ||||||
8. | ALA1258659 | 4-3 | t1/2 | = | 26.9 | min | ALA2379912 | hr | Rattus norvegicus | |||
9. | ALA1258659 | 4-3 | CLH | = | 85.8 | microL/min/mg | ALA2379913 | mL.min-1.g-1 | Rattus norvegicus | |||
10. | ALA1258659 | 4-3 | IC50 | = | 3.6 | uM | ALA1259549 | 5.44 | nM | Homo sapiens | ||
11. | ALA1258659 | 4-3 | IC50 | = | 0.7 | uM | ALA1259548 | 6.16 | nM | Homo sapiens |