# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1269411 | 2-HDA | CMC | > | 90 | ug ml-1 | ALA3362584 | ug ml-1 | ||||
2. | ALA1269411 | 2-HDA | MTD | = | 0.8 | uM | ALA3362582 | uM | Danio rerio | |||
3. | ALA1269411 | 2-HDA | IC50 | = | 85.9 | ug ml-1 | ALA3362581 | ug.mL-1 | Rattus norvegicus | |||
4. | ALA1269411 | 2-HDA | IC50 | = | 10.4 | ug ml-1 | ALA3362580 | ug.mL-1 | Plasmodium falciparum | |||
5. | ALA1269411 | 2-HDA | IC50 | = | 3.5 | ug ml-1 | ALA3362579 | ug.mL-1 | ||||
6. | ALA1269411 | 2-HDA | IC50 | = | 0.58 | ug ml-1 | ALA3362578 | ug.mL-1 | ||||
7. | ALA1269411 | 2-HDA | IC50 | = | 0.38 | ug ml-1 | ALA3362577 | ug.mL-1 | ||||
8. | ALA1269411 | 2-HDA | IC50 | = | 0.48 | ug ml-1 | ALA3362208 | ug.mL-1 | Plasmodium berghei | |||
9. | ALA1269411 | 2-HDA | INH | 0 | ALA2155871 | Not Active | % | |||||
10. | ALA1269411 | 2-HDA | INH | 0 | ALA2155884 | Active | % | Leishmania major | ||||
11. | ALA1269411 | 2-HDA | INH | 0 | ALA2155882 | Active | % | Leishmania major | ||||
12. | ALA1269411 | 2-HDA | IC50 | > | 100 | uM | ALA2155881 | nM | ||||
13. | ALA1269411 | 2-HDA | EC50 | > | 100 | uM | ALA2155880 | nM | ||||
14. | ALA1269411 | 2-HDA | EC50 | = | 28.7 | uM | ALA2155879 | 4.54 | nM | Leishmania major | ||
15. | ALA1269411 | 2-HDA | Activity | = | 2.77 | % | ALA2155878 | % | Leishmania infantum | |||
16. | ALA1269411 | 2-HDA | IC50 | = | 14.9 | uM | ALA2155877 | 4.83 | nM | Leishmania infantum | ||
17. | ALA1269411 | 2-HDA | IC50 | = | 340.3 | uM | ALA2155876 | nM | Rattus norvegicus | |||
18. | ALA1269411 | 2-HDA | IC50 | = | 17.8 | uM | ALA2155875 | 4.75 | nM | Leishmania donovani | ||
19. | ALA1269411 | 2-HDA | IC50 | = | 80 | uM | ALA2155874 | 4.10 | nM | Trypanosoma cruzi | ||
20. | ALA1269411 | 2-HDA | IC50 | = | 83.6 | uM | ALA2155873 | 4.08 | nM | Trypanosoma brucei rhodesiense |