# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1276947 | 64 | pKi | = | 7.5 | ALA1287093 | 7.50 | nM | Homo sapiens | |||
2. | ALA1276947 | 64 | pKi | = | 7.5 | ALA1287094 | 7.50 | nM | Homo sapiens | |||
3. | ALA1276947 | 64 | pKi | = | 6.4 | ALA1287095 | 6.40 | nM | Homo sapiens | |||
4. | ALA1276947 | 64 | pKi | = | 7.2 | ALA1287096 | 7.20 | nM | Homo sapiens | |||
5. | ALA1276947 | 64 | pKi | = | 8.27 | ALA1287099 | 8.27 | nM | Rattus norvegicus | |||
6. | ALA1276947 | 64 | pKi | = | 7.16 | ALA1287100 | 7.16 | nM | Rattus norvegicus | |||
7. | ALA1276947 | 64 | pIC50 | < | 4.4 | ALA1287098 | nM | Homo sapiens | ||||
8. | ALA1276947 | 64 | CL | < | 0.5 | ml/min/g | ALA1287101 | mL.min-1.g-1 | Rattus norvegicus | |||
9. | ALA1276947 | 64 | CL | < | 0.5 | ml/min/g | ALA1287102 | mL.min-1.g-1 | Homo sapiens | |||
10. | ALA1276947 | 64 | IC50 | > | 10 | uM | ALA1287103 | nM | Homo sapiens | |||
11. | ALA1276947 | 64 | IC50 | > | 10 | uM | ALA1287104 | nM | Homo sapiens | |||
12. | ALA1276947 | 64 | IC50 | > | 10 | uM | ALA1287105 | nM | Homo sapiens | |||
13. | ALA1276947 | 64 | IC50 | > | 10 | uM | ALA1287106 | nM | Homo sapiens | |||
14. | ALA1276947 | 64 | IC50 | > | 10 | uM | ALA1287107 | nM | Homo sapiens | |||
15. | ALA1276947 | 64 | Fu | = | 2.3 | % | ALA1287108 | Rattus norvegicus | ||||
16. | ALA1276947 | 64 | Fu | = | 8 | % | ALA1287109 | Rattus norvegicus | ||||
17. | ALA1276947 | 64 | CL | = | 5 | ml/min.kg | ALA1287110 | mL.min-1.kg-1 | Rattus norvegicus | |||
18. | ALA1276947 | 64 | Vdss | = | 2.4 | L/Kg | ALA1287112 | L.kg-1 | Rattus norvegicus | |||
19. | ALA1276947 | 64 | t1/2 | = | 5.3 | hr | ALA1287114 | hr | Rattus norvegicus | |||
20. | ALA1276947 | 64 | F | = | 62 | % | ALA1287116 | % | Rattus norvegicus |