# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1277126 | 69 | CL | = | 16 | ml/min.kg | ALA1287111 | mL.min-1.kg-1 | Rattus norvegicus | |||
2. | ALA1277126 | 69 | pKi | = | 7.3 | ALA1287093 | 7.30 | nM | Homo sapiens | |||
3. | ALA1277126 | 69 | pKi | = | 7.6 | ALA1287094 | 7.60 | nM | Homo sapiens | |||
4. | ALA1277126 | 69 | pKi | < | 5.7 | ALA1287095 | nM | Homo sapiens | ||||
5. | ALA1277126 | 69 | pKi | = | 6 | ALA1287096 | 6.00 | nM | Homo sapiens | |||
6. | ALA1277126 | 69 | pKi | = | 7.7 | ALA1287099 | 7.70 | nM | Rattus norvegicus | |||
7. | ALA1277126 | 69 | pKi | = | 6.98 | ALA1287100 | 6.98 | nM | Rattus norvegicus | |||
8. | ALA1277126 | 69 | CL | < | 0.5 | ml/min/g | ALA1287101 | mL.min-1.g-1 | Rattus norvegicus | |||
9. | ALA1277126 | 69 | CL | < | 0.5 | ml/min/g | ALA1287102 | mL.min-1.g-1 | Homo sapiens | |||
10. | ALA1277126 | 69 | IC50 | > | 10 | uM | ALA1287103 | nM | Homo sapiens | |||
11. | ALA1277126 | 69 | IC50 | > | 10 | uM | ALA1287104 | nM | Homo sapiens | |||
12. | ALA1277126 | 69 | IC50 | > | 10 | uM | ALA1287105 | nM | Homo sapiens | |||
13. | ALA1277126 | 69 | IC50 | > | 10 | uM | ALA1287106 | nM | Homo sapiens | |||
14. | ALA1277126 | 69 | IC50 | > | 10 | uM | ALA1287107 | nM | Homo sapiens | |||
15. | ALA1277126 | 69 | Fu | = | 2.7 | % | ALA1287108 | Rattus norvegicus | ||||
16. | ALA1277126 | 69 | Fu | = | 10.3 | % | ALA1287109 | Rattus norvegicus | ||||
17. | ALA1277126 | 69 | Vdss | = | 2.7 | L/Kg | ALA1287113 | L.kg-1 | Rattus norvegicus | |||
18. | ALA1277126 | 69 | t1/2 | = | 3 | hr | ALA1287115 | hr | Rattus norvegicus | |||
19. | ALA1277126 | 69 | F | = | 37 | % | ALA1287117 | % | Rattus norvegicus | |||
20. | ALA1277126 | 69 | BBR | = | 1.8 | ALA1287119 |