# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1289827 | NSC-748393 | CC50 | = | 10 | uM | ALA2090698 | nM | Chlorocebus sabaeus | |||
2. | ALA1289827 | NSC-748393 | Ratio CC50/IC50 | = | 333 | ALA2090699 | ||||||
3. | ALA1289827 | NSC-748393 | IC50 | = | 0.03 | uM | ALA2090694 | 7.52 | nM | Trypanosoma brucei brucei | ||
4. | ALA1289827 | NSC-748393 | IC50 | = | 22 | uM | ALA2090695 | 4.66 | nM | |||
5. | ALA1289827 | NSC-748393 | IC50 | = | 55 | uM | ALA2090696 | 4.26 | nM | Trypanosoma brucei | ||
6. | ALA1289827 | NSC-748393 | IC50 | = | 6 | uM | ALA2090697 | 5.22 | nM | Trypanosoma brucei rhodesiense | ||
7. | ALA1289827 | NSC-748393 | Ratio | = | 1.6 | ALA1292269 | ||||||
8. | ALA1289827 | NSC-748393 | deltaTm | = | 13.1 | degrees C | ALA1292268 | degrees C | ||||
9. | ALA1289827 | NSC-748393 | deltaTm | = | 20.9 | degrees C | ALA1292267 | degrees C | ||||
10. | ALA1289827 | NSC-748393 | MTD | = | 50 | mg kg-1 | ALA1292266 | mg kg-1 | Mus musculus | |||
11. | ALA1289827 | NSC-748393 | pLC50 | = | 5.67 | ALA1292265 | nM | Homo sapiens | ||||
12. | ALA1289827 | NSC-748393 | pLC50 | = | 4.59 | ALA1292264 | nM | Homo sapiens | ||||
13. | ALA1289827 | NSC-748393 | pLC50 | = | 5.1 | ALA1292263 | nM | Homo sapiens | ||||
14. | ALA1289827 | NSC-748393 | pLC50 | = | 5.25 | ALA1293174 | nM | Homo sapiens | ||||
15. | ALA1289827 | NSC-748393 | pLC50 | = | 4.03 | ALA1293175 | nM | |||||
16. | ALA1289827 | NSC-748393 | pLC50 | = | 4 | ALA1293176 | nM | Homo sapiens | ||||
17. | ALA1289827 | NSC-748393 | pLC50 | > | 4 | ALA1293177 | nM | Homo sapiens | ||||
18. | ALA1289827 | NSC-748393 | pLC50 | > | 4.44 | ALA1293178 | nM | Homo sapiens | ||||
19. | ALA1289827 | NSC-748393 | pLC50 | = | 4.05 | ALA1293179 | nM | Homo sapiens | ||||
20. | ALA1289827 | NSC-748393 | pLC50 | = | 4 | ALA1293180 | nM | Homo sapiens |