# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1289828 | NSC-748394 | IC50 | = | 1 | uM | ALA2090697 | 6.00 | nM | Trypanosoma brucei rhodesiense | ||
2. | ALA1289828 | NSC-748394 | CC50 | = | 4.8 | uM | ALA2090698 | nM | Chlorocebus sabaeus | |||
3. | ALA1289828 | NSC-748394 | Ratio CC50/IC50 | = | 60 | ALA2090699 | ||||||
4. | ALA1289828 | NSC-748394 | IC50 | = | 0.08 | uM | ALA2090694 | 7.10 | nM | Trypanosoma brucei brucei | ||
5. | ALA1289828 | NSC-748394 | IC50 | = | 3 | uM | ALA2090695 | 5.52 | nM | |||
6. | ALA1289828 | NSC-748394 | IC50 | = | 76 | uM | ALA2090696 | 4.12 | nM | Trypanosoma brucei | ||
7. | ALA1289828 | NSC-748394 | Ratio | = | 4 | ALA1292269 | ||||||
8. | ALA1289828 | NSC-748394 | deltaTm | = | 1.2 | degrees C | ALA1292268 | degrees C | ||||
9. | ALA1289828 | NSC-748394 | deltaTm | = | 4.2 | degrees C | ALA1292267 | degrees C | ||||
10. | ALA1289828 | NSC-748394 | MTD | = | 160 | mg kg-1 | ALA1292266 | mg kg-1 | Mus musculus | |||
11. | ALA1289828 | NSC-748394 | pLC50 | = | 6.05 | ALA1292265 | nM | Homo sapiens | ||||
12. | ALA1289828 | NSC-748394 | pLC50 | = | 5.28 | ALA1292263 | nM | Homo sapiens | ||||
13. | ALA1289828 | NSC-748394 | pLC50 | = | 5.31 | ALA1293174 | nM | Homo sapiens | ||||
14. | ALA1289828 | NSC-748394 | pLC50 | = | 5.22 | ALA1293176 | nM | Homo sapiens | ||||
15. | ALA1289828 | NSC-748394 | pLC50 | = | 6.04 | ALA1293178 | nM | Homo sapiens | ||||
16. | ALA1289828 | NSC-748394 | pLC50 | = | 5.38 | ALA1293179 | nM | Homo sapiens | ||||
17. | ALA1289828 | NSC-748394 | pLC50 | = | 5.49 | ALA1293180 | nM | Homo sapiens | ||||
18. | ALA1289828 | NSC-748394 | pLC50 | = | 5.52 | ALA1293181 | nM | Homo sapiens | ||||
19. | ALA1289828 | NSC-748394 | pLC50 | = | 5.25 | ALA1293182 | nM | Homo sapiens | ||||
20. | ALA1289828 | NSC-748394 | pLC50 | = | 5.17 | ALA1293183 | nM | Homo sapiens |