# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1290717 | SI R18C1 | IC50 | = | 2 | uM | ALA2090697 | 5.70 | nM | Trypanosoma brucei rhodesiense | ||
2. | ALA1290717 | SI R18C1 | CC50 | = | 2.6 | uM | ALA2090698 | nM | Chlorocebus sabaeus | |||
3. | ALA1290717 | SI R18C1 | Ratio CC50/IC50 | = | 8.6 | ALA2090699 | ||||||
4. | ALA1290717 | SI R18C1 | IC50 | = | 0.3 | uM | ALA2090694 | 6.52 | nM | Trypanosoma brucei brucei | ||
5. | ALA1290717 | SI R18C1 | IC50 | = | 5 | uM | ALA2090695 | 5.30 | nM | |||
6. | ALA1290717 | SI R18C1 | IC50 | = | 59 | uM | ALA2090696 | 4.23 | nM | Trypanosoma brucei | ||
7. | ALA1290717 | SI R18C1 | Ka | = | 1 | 10'6/M | ALA1681229 | 10'6/M | ||||
8. | ALA1290717 | SI R18C1 | IC50 | 0 | ALA1681231 | Not Determined | ||||||
9. | ALA1290717 | SI R18C1 | IC50 | = | 9.32 | uM | ALA1681230 | 5.03 | nM | |||
10. | ALA1290717 | SI R18C1 | Ka | = | 0.17 | 10'6/M | ALA1681228 | 10'6/M | ||||
11. | ALA1290717 | SI R18C1 | Ratio IC50 | = | 0.6 | ALA1681221 | Plasmodium falciparum | |||||
12. | ALA1290717 | SI R18C1 | Ratio IC50 | = | 14 | ALA1681220 | ||||||
13. | ALA1290717 | SI R18C1 | IC50 | = | 2.6 | uM | ALA1681219 | 5.58 | nM | Chlorocebus sabaeus | ||
14. | ALA1290717 | SI R18C1 | IC50 | = | 166 | nM | ALA1681218 | 6.78 | nM | Plasmodium falciparum | ||
15. | ALA1290717 | SI R18C1 | IC50 | = | 279 | nM | ALA1681217 | 6.55 | nM | Plasmodium falciparum | ||
16. | ALA1290717 | SI R18C1 | IC50 | = | 247 | nM | ALA1681216 | 6.61 | nM | Plasmodium falciparum | ||
17. | ALA1290717 | SI R18C1 | IC50 | = | 180 | nM | ALA1681215 | 6.75 | nM | Plasmodium falciparum | ||
18. | ALA1290717 | SI R18C1 | pKa | = | 10.3 | ALA1292260 | ||||||
19. | ALA1290717 | SI R18C1 | IC50 | = | 2.6 | uM | ALA1292262 | 5.58 | nM | Chlorocebus sabaeus |