| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1405739 | SID49645185 | IC50_Mean | > | 66 | uM | ALA1963941 | inactive | nM | Homo sapiens | ||
| 2. | ALA1405739 | SID49645185 | Potency | 14.125 | uM | ALA2114916 | inconclusive | nM | Trypanosoma brucei brucei (strain 927/4 GUTat10.1) | |||
| 3. | ALA1405739 | SID49645185 | Potency | 15.849 | uM | ALA2114913 | inconclusive | nM | Homo sapiens | |||
| 4. | ALA1405739 | SID49645185 | Potency | 26.68 | uM | ALA3215278 | active | nM | Homo sapiens | |||
| 5. | ALA1405739 | SID49645185 | pIC50 | = | 7.01 | ALA3424956 | 7.01 | nM | Rattus norvegicus | |||
| 6. | ALA1405739 | SID49645185 | INH | 0 | ALA3424972 | Dose-dependent effect | % | Rattus norvegicus | ||||
| 7. | ALA1405739 | SID49645185 | Activity | = | 395.06 | nmol/g | ALA3424971 | nmol/g | Rattus norvegicus | |||
| 8. | ALA1405739 | SID49645185 | Activity | = | 478.71 | nmol/g | ALA3424970 | nmol/g | Rattus norvegicus | |||
| 9. | ALA1405739 | SID49645185 | Activity | = | 536.01 | nmol/g | ALA3424968 | nmol/g | Rattus norvegicus | |||
| 10. | ALA1405739 | SID49645185 | Activity | = | 668.66 | nmol/g | ALA3424969 | nmol/g | Rattus norvegicus | |||
| 11. | ALA1405739 | SID49645185 | logD | = | -1.9 | ALA3424967 | ||||||
| 12. | ALA1405739 | SID49645185 | Ki | = | 0.089 | umol/L | ALA3424966 | 7.05 | nM | Rattus norvegicus | ||
| 13. | ALA1405739 | SID49645185 | Ratio IC50 | > | 200 | ALA3424965 | ||||||
| 14. | ALA1405739 | SID49645185 | IC50 | = | 21.4 | uM | ALA3424964 | 4.67 | nM | Homo sapiens | ||
| 15. | ALA1405739 | SID49645185 | Ratio IC50 | > | 400 | ALA3424963 | ||||||
| 16. | ALA1405739 | SID49645185 | IC50 | = | 0.057 | uM | ALA3424962 | 7.24 | nM | Homo sapiens | ||
| 17. | ALA1405739 | SID49645185 | IC50 | = | 0.097 | uM | ALA3424956 | 7.01 | nM | Rattus norvegicus | ||
| 18. | ALA1405739 | SID49645185 | IC50 | = | 40.55 | uM | ALA3424959 | 4.39 | nM | Rattus norvegicus | ||
| 19. | ALA1405739 | SID49645185 | Potency | 25.119 | uM | ALA1614166 | inconclusive | nM | Homo sapiens | |||
| 20. | ALA1405739 | SID49645185 | Potency | 10 | uM | ALA3215181 | inactive | nM |
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