| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA11081 | 1a (UH5) | Inhibition | = | 100 | % | ALA663185 | % | Rattus norvegicus | |||
| 2. | ALA11081 | 1a (UH5) | PI turnover | = | 41.6 | ALA619660 | Mus musculus | |||||
| 3. | ALA11081 | 1a (UH5) | PI turnover | = | 52.5 | ALA619657 | Mus musculus | |||||
| 4. | ALA11081 | 1a (UH5) | Displacement | = | 94.7 | % | ALA748794 | % | Rattus norvegicus | |||
| 5. | ALA11081 | 1a (UH5) | Displacement | = | 89.4 | % | ALA749278 | % | Rattus norvegicus | |||
| 6. | ALA11081 | 1a (UH5) | Relative efficacy | = | 0.15 | ALA688026 | Cavia porcellus | |||||
| 7. | ALA11081 | 1a (UH5) | Kd | = | 2.2 | uM | ALA686995 | 5.66 | nM | Homo sapiens | ||
| 8. | ALA11081 | 1a (UH5) | Emax | = | 1.01 | ALA692167 | Cavia porcellus | |||||
| 9. | ALA11081 | 1a (UH5) | EC50 | = | 0.069 | uM | ALA684549 | 7.16 | nM | Cavia porcellus | ||
| 10. | ALA11081 | 1a (UH5) | Selectivity ratio | = | 0.9 | ALA839035 | ||||||
| 11. | ALA11081 | 1a (UH5) | IC50 | = | 2450 | nM | ALA745679 | 5.61 | nM | Homo sapiens | ||
| 12. | ALA11081 | 1a (UH5) | IC50 | = | 2010 | nM | ALA744023 | 5.70 | nM | Rattus norvegicus | ||
| 13. | ALA11081 | 1a (UH5) | Efficacy ratio | = | 544 | ALA882585 | Rattus norvegicus | |||||
| 14. | ALA11081 | 1a (UH5) | IC50 | = | 2447 | nM | ALA748213 | 5.61 | nM | Rattus norvegicus | ||
| 15. | ALA11081 | 1a (UH5) | IC50 | = | 4.5 | nM | ALA748432 | 8.35 | nM | Rattus norvegicus | ||
| 16. | ALA11081 | 1a (UH5) | Ki | = | 4.96 | uM | ALA749269 | 5.30 | nM | Homo sapiens | ||
| 17. | ALA11081 | 1a (UH5) | Ki | = | 4.5 | uM | ALA745460 | 5.35 | nM | Rattus norvegicus | ||
| 18. | ALA11081 | 1a (UH5) | Affinity | = | 88.8 | % | ALA744388 | % | Homo sapiens | |||
| 19. | ALA11081 | 1a (UH5) | Activity | = | 48 | % | ALA745522 | % | Homo sapiens | |||
| 20. | ALA11081 | 1a (UH5) | Affinity | = | 79.6 | % | ALA745068 | % | Rattus norvegicus |
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