# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1422005 | SID26729800 | Kd | = | 1.8 | uM | ALA4419254 | 5.75 | nM | Homo sapiens | ||
2. | ALA1422005 | SID26729800 | INH | 0 | ALA4419294 | Active | % | Homo sapiens | ||||
3. | ALA1422005 | SID26729800 | INH | 0 | ALA4419293 | Active | % | Homo sapiens | ||||
4. | ALA1422005 | SID26729800 | INH | 0 | ALA4419292 | Active | % | Homo sapiens | ||||
5. | ALA1422005 | SID26729800 | INH | 0 | ALA4419291 | Active | % | Homo sapiens | ||||
6. | ALA1422005 | SID26729800 | RUmax | = | 0.761 | 10'2/Da | ALA4419290 | 10'2/Da | Homo sapiens | |||
7. | ALA1422005 | SID26729800 | RUmax | = | 0.205 | 10'2/Da | ALA4419289 | 10'2/Da | Homo sapiens | |||
8. | ALA1422005 | SID26729800 | IC50 | > | 100 | uM | ALA4419288 | nM | Homo sapiens | |||
9. | ALA1422005 | SID26729800 | IC50 | = | 15 | uM | ALA4419287 | 4.82 | nM | Homo sapiens | ||
10. | ALA1422005 | SID26729800 | beta t1/2 | = | 3 | min | ALA4419253 | hr | ||||
11. | ALA1422005 | SID26729800 | t1/2 | = | 99 | min | ALA4419284 | hr | Homo sapiens | |||
12. | ALA1422005 | SID26729800 | t1/2 | = | 19 | min | ALA4419283 | hr | Homo sapiens | |||
13. | ALA1422005 | SID26729800 | t1/2 | = | 790 | min | ALA4419282 | hr | ||||
14. | ALA1422005 | SID26729800 | t1/2 | 0 | ALA4419281 | Stable | ||||||
15. | ALA1422005 | SID26729800 | t1/2 | = | 558 | min | ALA4419280 | hr | ||||
16. | ALA1422005 | SID26729800 | t1/2 | = | 6.3 | min | ALA4419279 | hr | ||||
17. | ALA1422005 | SID26729800 | IC50 | = | 70 | uM | ALA4419278 | 4.16 | nM | Homo sapiens | ||
18. | ALA1422005 | SID26729800 | IC50 | = | 27 | uM | ALA4419277 | 4.57 | nM | Homo sapiens | ||
19. | ALA1422005 | SID26729800 | IC50 | = | 51 | uM | ALA4419276 | 4.29 | nM | |||
20. | ALA1422005 | SID26729800 | IC50 | > | 100 | uM | ALA4419275 | nM | Homo sapiens |