| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA428848 | 13b | F | = | 88 | % | ALA5150514 | % | ||||
| 2. | ALA428848 | 13b | F | = | 62 | % | ALA5150513 | % | ||||
| 3. | ALA428848 | 13b | F | = | 77 | % | ALA5150512 | % | ||||
| 4. | ALA428848 | 13b | ED50 | = | 7.5 | mg kg-1 | ALA4399456 | mg.kg-1 | Cricetinae | |||
| 5. | ALA428848 | 13b | F | = | 88 | % | ALA4399452 | % | ||||
| 6. | ALA428848 | 13b | F | = | 62 | % | ALA4399451 | % | ||||
| 7. | ALA428848 | 13b | Ki | = | 101 | nM | ALA4399449 | 7.00 | nM | Homo sapiens | ||
| 8. | ALA428848 | 13b | LogD7.4 | 1.05 | ALA3301363 | |||||||
| 9. | ALA428848 | 13b | ED50 | = | 7.5 | mg kg-1 | ALA690251 | mg.kg-1 | Cricetinae gen. sp. | |||
| 10. | ALA428848 | 13b | Ki | = | 101 | nM | ALA677434 | 7.00 | nM | Homo sapiens | ||
| 11. | ALA428848 | 13b | Bioavailabiility | = | 88 | % | ALA620562 | % | Canis lupus familiaris | |||
| 12. | ALA428848 | 13b | AUC | = | 357 | min ug ml-1 | ALA621081 | ng.hr.mL-1 | Canis lupus familiaris | |||
| 13. | ALA428848 | 13b | T max | = | 60 | min | ALA635770 | hr | Canis lupus familiaris | |||
| 14. | ALA428848 | 13b | Cmax | = | 3.23 | ug ml-1 | ALA626037 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Canis lupus familiaris | ||
| 15. | ALA428848 | 13b | T1/2 | = | 58 | min | ALA858570 | hr | Canis lupus familiaris | |||
| 16. | ALA428848 | 13b | Bioavailabiility | = | 62 | % | ALA620564 | % | Rattus norvegicus | |||
| 17. | ALA428848 | 13b | AUC | = | 310 | min ug ml-1 | ALA621083 | ng.hr.mL-1 | Rattus norvegicus | |||
| 18. | ALA428848 | 13b | T max | = | 60 | min | ALA633558 | hr | ||||
| 19. | ALA428848 | 13b | Cmax | = | 1.9 | ug ml-1 | ALA626039 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 20. | ALA428848 | 13b | T1/2 | = | 96 | min | ALA873838 | hr | Rattus norvegicus |
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