# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Imatinib (STI571) | 1 | IC50 | = | 16.59 | uM | ALA5249271 | 4.78 | nM | Homo sapiens | ||
2. | Imatinib (STI571) | 1 | IC50 | = | 28.54 | uM | ALA5249270 | 4.54 | nM | Homo sapiens | ||
3. | Imatinib (STI571) | 1 | IC50 | = | 0.135 | uM | ALA5249269 | 6.87 | nM | Homo sapiens | ||
4. | Imatinib (STI571) | 1 | solubility | = | 30.7 | uM | ALA5247282 | nM | ||||
5. | Imatinib (STI571) | 1 | IC50 | = | 0.37 | uM | ALA5247281 | 6.43 | nM | Homo sapiens | ||
6. | Imatinib (STI571) | 1 | IC50 | > | 100 | uM | ALA5244903 | nM | Homo sapiens | |||
7. | Imatinib (STI571) | 1 | IC50 | = | 50 | nM | ALA5244902 | 7.30 | nM | Mus musculus | ||
8. | Imatinib (STI571) | 1 | IC50 | = | 38 | nM | ALA5244901 | 7.42 | nM | Mus musculus | ||
9. | Imatinib (STI571) | 1 | Activity | = | 23.1 | % | ALA5241030 | % | Homo sapiens | |||
10. | Imatinib (STI571) | 1 | Activity | = | 0.2 | % | ALA5241029 | % | Homo sapiens | |||
11. | Imatinib (STI571) | 1 | Activity | = | 18.2 | % | ALA5241028 | % | Homo sapiens | |||
12. | Imatinib (STI571) | 1 | Activity | = | 4.9 | % | ALA5241027 | % | Homo sapiens | |||
13. | Imatinib (STI571) | 1 | Activity | = | 76.7 | % | ALA5241026 | % | Homo sapiens | |||
14. | Imatinib (STI571) | 1 | IC50 | = | 25.55 | uM | ALA5241016 | 4.59 | nM | Homo sapiens | ||
15. | Imatinib (STI571) | 1 | IC50 | = | 17.2 | uM | ALA5241015 | 4.76 | nM | Homo sapiens | ||
16. | Imatinib (STI571) | 1 | IC50 | = | 13.97 | uM | ALA5241014 | 4.86 | nM | Homo sapiens | ||
17. | Imatinib (STI571) | 1 | IC50 | >= | 6400 | nM | ALA5237471 | nM | Homo sapiens | |||
18. | Imatinib (STI571) | 1 | IC50 | = | 260 | nM | ALA5237470 | 6.58 | nM | Homo sapiens | ||
19. | Imatinib (STI571) | 1 | PPB | = | 95 | % | ALA5233776 | % | ||||
20. | Imatinib (STI571) | 1 | AUC | = | 24.8 | mg/L.hr | ALA5233773 | ng.hr.mL-1 |