| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA301018 | 4 | IC50 | = | 5300 | nM | ALA3631056 | 5.28 | nM | Homo sapiens | ||
| 2. | ALA301018 | 4 | IC50 | = | 400 | nM | ALA3631055 | 6.40 | nM | Homo sapiens | ||
| 3. | ALA301018 | 4 | Cmax | = | 7441 | ng/ml | ALA5226163 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 4. | ALA301018 | 4 | AUC | = | 26281 | ng.hr/ml | ALA5226161 | ng.hr.mL-1 | ||||
| 5. | ALA301018 | 4 | AUCt | = | 25480 | ng.hr/ml | ALA5226159 | ng.hr.mL-1 | ||||
| 6. | ALA301018 | 4 | beta t1/2 | = | 1.9 | hr | ALA5226157 | hr | ||||
| 7. | ALA301018 | 4 | solubility | = | 63.88 | ug ml-1 | ALA5226155 | ug.mL-1 | ||||
| 8. | ALA301018 | 4 | solubility | = | 51.72 | ug ml-1 | ALA5226154 | ug.mL-1 | ||||
| 9. | ALA301018 | 4 | solubility | = | 23.61 | ug ml-1 | ALA5226153 | ug.mL-1 | ||||
| 10. | ALA301018 | 4 | solubility | = | 49.42 | ug ml-1 | ALA5226152 | ug.mL-1 | ||||
| 11. | ALA301018 | 4 | solubility | = | 1.53 | ug ml-1 | ALA5226151 | ug.mL-1 | ||||
| 12. | ALA301018 | 4 | solubility | = | 1.3 | ug ml-1 | ALA5226150 | ug.mL-1 | ||||
| 13. | ALA301018 | 4 | pKa | = | 4.51 | ALA5226149 | ||||||
| 14. | ALA301018 | 4 | IC50 | = | 9 | nM | ALA5226148 | 8.05 | nM | Homo sapiens | ||
| 15. | ALA301018 | 4 | Solubility | 7.2 | uM | ALA3301364 | nM | |||||
| 16. | ALA301018 | 4 | LogD7.4 | 3.67 | ALA3301363 | |||||||
| 17. | ALA301018 | 4 | IC50 | = | 23 | nM | ALA4233281 | 7.64 | nM | Homo sapiens | ||
| 18. | ALA301018 | 4 | IC50 | = | 3.8 | nM | ALA2341281 | 8.42 | nM | Homo sapiens | ||
| 19. | ALA301018 | 4 | IC50 | = | 9 | nM | ALA2341279 | 8.05 | nM | Homo sapiens | ||
| 20. | ALA301018 | 4 | IC50 | = | 4.9 | uM | ALA2020646 | 5.31 | nM | Homo sapiens |
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