# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA301018 | 4 | IC50 | = | 3.8 | nM | ALA2341281 | 8.42 | nM | Homo sapiens | ||
2. | ALA301018 | 4 | IC50 | = | 9 | nM | ALA2341279 | 8.05 | nM | Homo sapiens | ||
3. | ALA301018 | 4 | IC50 | = | 4.9 | uM | ALA2020646 | 5.31 | nM | Homo sapiens | ||
4. | ALA301018 | 4 | IC50 | = | 5.7 | uM | ALA2020645 | 5.24 | nM | Homo sapiens | ||
5. | ALA301018 | 4 | IC50 | = | 6.5 | uM | ALA2020644 | 5.19 | nM | Homo sapiens | ||
6. | ALA301018 | 4 | IC50 | = | 5.3 | uM | ALA2020643 | 5.28 | nM | Homo sapiens | ||
7. | ALA301018 | 4 | IC50 | = | 0.38 | uM | ALA2020642 | 6.42 | nM | Homo sapiens | ||
8. | ALA301018 | 4 | Solubility | 7.2 | uM | ALA3301364 | nM | |||||
9. | ALA301018 | 4 | LogD7.4 | 3.67 | ALA3301363 | |||||||
10. | ALA301018 | 4 | IC50 | = | 23 | nM | ALA4233281 | 7.64 | nM | Homo sapiens | ||
11. | ALA301018 | 4 | IC50 | = | 0.29 | uM | ALA5263443 | 6.54 | nM | Homo sapiens | ||
12. | ALA301018 | 4 | Cmax | = | 7441 | ng/ml | ALA5226163 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
13. | ALA301018 | 4 | AUC | = | 26281 | ng.hr/ml | ALA5226161 | ng.hr.mL-1 | ||||
14. | ALA301018 | 4 | AUCt | = | 25480 | ng.hr/ml | ALA5226159 | ng.hr.mL-1 | ||||
15. | ALA301018 | 4 | beta t1/2 | = | 1.9 | hr | ALA5226157 | hr | ||||
16. | ALA301018 | 4 | solubility | = | 63.88 | ug ml-1 | ALA5226155 | ug.mL-1 | ||||
17. | ALA301018 | 4 | solubility | = | 51.72 | ug ml-1 | ALA5226154 | ug.mL-1 | ||||
18. | ALA301018 | 4 | solubility | = | 23.61 | ug ml-1 | ALA5226153 | ug.mL-1 | ||||
19. | ALA301018 | 4 | solubility | = | 49.42 | ug ml-1 | ALA5226152 | ug.mL-1 | ||||
20. | ALA301018 | 4 | solubility | = | 1.53 | ug ml-1 | ALA5226151 | ug.mL-1 |