# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA292521 | 5 | ED50 | > | 100 | mg kg-1 | ALA5236049 | mg.kg-1 | Mus musculus | |||
2. | ALA292521 | 5 | INH | 0 | ALA5236048 | Not Active | % | Mus musculus | ||||
3. | ALA292521 | 5 | Emax | = | 87 | % | ALA5236047 | % | Mus musculus | |||
4. | ALA292521 | 5 | EC50 | = | 857.8 | nM | ALA5236046 | 6.07 | nM | Mus musculus | ||
5. | ALA292521 | 5 | Emax | = | 62 | % | ALA5236042 | % | Mus musculus | |||
6. | ALA292521 | 5 | EC50 | = | 422.4 | nM | ALA5236041 | 6.37 | nM | Mus musculus | ||
7. | ALA292521 | 5 | Ki | = | 1882.4 | nM | ALA5236040 | 5.72 | nM | Mus musculus | ||
8. | ALA292521 | 5 | Ki | = | 1177.2 | nM | ALA5236039 | 5.93 | nM | Mus musculus | ||
9. | ALA292521 | 5 | Ki | = | 216.2 | nM | ALA5236038 | 6.67 | nM | Mus musculus | ||
10. | ALA292521 | 5 | Ki | = | 105 | nM | ALA4380084 | 6.98 | nM | Homo sapiens | ||
11. | ALA292521 | 5 | Ki | 0 | ALA4380083 | Not Determined | Homo sapiens | |||||
12. | ALA292521 | 5 | Ki | 0 | ALA4380082 | Not Determined | Homo sapiens | |||||
13. | ALA292521 | 5 | INH | = | 28.9 | % | ALA4380081 | % | Homo sapiens | |||
14. | ALA292521 | 5 | INH | = | 95.4 | % | ALA4380080 | % | Homo sapiens | |||
15. | ALA292521 | 5 | INH | = | 39.5 | % | ALA4380079 | % | Homo sapiens | |||
16. | ALA292521 | 5 | INH | = | 25.3 | % | ALA4380078 | % | Homo sapiens | |||
17. | ALA292521 | 5 | INH | = | 14.6 | % | ALA4380077 | % | Homo sapiens | |||
18. | ALA292521 | 5 | INH | = | 20 | % | ALA4380076 | % | Homo sapiens | |||
19. | ALA292521 | 5 | INH | = | 66.3 | % | ALA4380075 | % | Homo sapiens | |||
20. | ALA292521 | 5 | INH | = | 29 | % | ALA4380074 | % | Homo sapiens |