| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA59765 | 28 | PB | = | 94 | % | ALA977256 | % | Canis lupus familiaris | |||
| 2. | ALA59765 | 28 | INH | = | 40.8 | % | ALA977255 | % | Canis lupus familiaris | |||
| 3. | ALA59765 | 28 | EC50 | = | 30 | nM | ALA977254 | 7.52 | nM | Canis lupus familiaris | ||
| 4. | ALA59765 | 28 | F | = | 29 | % | ALA977244 | % | Rattus norvegicus | |||
| 5. | ALA59765 | 28 | F | = | 73 | % | ALA977247 | % | Canis lupus familiaris | |||
| 6. | ALA59765 | 28 | F | = | 35 | % | ALA977250 | % | Macaca mulatta | |||
| 7. | ALA59765 | 28 | CL | = | 11.8 | ml/min.kg | ALA977249 | mL.min-1.kg-1 | Macaca mulatta | |||
| 8. | ALA59765 | 28 | CL | = | 3.7 | ml/min.kg | ALA977246 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 9. | ALA59765 | 28 | CL | = | 47.9 | ml/min.kg | ALA977243 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 10. | ALA59765 | 28 | t1/2 | = | 2.28 | hr | ALA977248 | hr | Macaca mulatta | |||
| 11. | ALA59765 | 28 | t1/2 | = | 1.63 | hr | ALA977245 | hr | Canis lupus familiaris | |||
| 12. | ALA59765 | 28 | t1/2 | = | 0.3 | hr | ALA977242 | hr | Rattus norvegicus | |||
| 13. | ALA59765 | 28 | AUC | = | 4100 | ng.hr/ml | ALA976376 | ng.hr.mL-1 | Homo sapiens | |||
| 14. | ALA59765 | 28 | AUC | = | 398 | ng.hr/ml | ALA976364 | ng.hr.mL-1 | Macaca mulatta | |||
| 15. | ALA59765 | 28 | AUC | = | 10600 | ng.hr/ml | ALA976374 | ng.hr.mL-1 | Canis lupus familiaris | |||
| 16. | ALA59765 | 28 | AUC | = | 83 | ng.hr/ml | ALA976368 | ng.hr.mL-1 | Rattus norvegicus | |||
| 17. | ALA59765 | 28 | Cmax | = | 1340 | ng/ml | ALA976375 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Homo sapiens | ||
| 18. | ALA59765 | 28 | Cmax | = | 184 | ng/ml | ALA976363 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Macaca mulatta | ||
| 19. | ALA59765 | 28 | Cmax | = | 2070 | ng/ml | ALA976373 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Canis lupus familiaris | ||
| 20. | ALA59765 | 28 | Cmax | = | 38 | ng/ml | ALA976367 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus |
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