| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA62811 | 19 | INH | < | 5 | % | ALA3399808 | % | Rattus norvegicus | |||
| 2. | ALA62811 | 19 | INH | = | 31 | % | ALA3399807 | % | Homo sapiens | |||
| 3. | ALA62811 | 19 | INH | = | 20 | % | ALA3399806 | % | Homo sapiens | |||
| 4. | ALA62811 | 19 | Ratio IC50 | = | 241 | ALA3399804 | ||||||
| 5. | ALA62811 | 19 | IC50 | = | 6746 | nM | ALA3399803 | 5.17 | nM | Homo sapiens | ||
| 6. | ALA62811 | 19 | IC50 | = | 28 | nM | ALA3399802 | 7.55 | nM | Homo sapiens | ||
| 7. | ALA62811 | 19 | IC50 | = | 28 | nM | ALA1768362 | 7.55 | nM | Homo sapiens | ||
| 8. | ALA62811 | 19 | IC50 | > | 5000 | nM | ALA2166348 | nM | Homo sapiens | |||
| 9. | ALA62811 | 19 | F | = | 71 | % | ALA990671 | % | Rattus norvegicus | |||
| 10. | ALA62811 | 19 | AUC | = | 270 | ng.hr/ml | ALA990670 | ng.hr.mL-1 | Rattus norvegicus | |||
| 11. | ALA62811 | 19 | AUC | = | 4762 | ng.hr/ml | ALA990669 | ng.hr.mL-1 | Rattus norvegicus | |||
| 12. | ALA62811 | 19 | Cmax | = | 1537 | ng/mL | ALA990667 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 13. | ALA62811 | 19 | Tmax | = | 1 | hr | ALA990665 | hr | Rattus norvegicus | |||
| 14. | ALA62811 | 19 | beta t1/2 | = | 1.7 | hr | ALA990663 | hr | Rattus norvegicus | |||
| 15. | ALA62811 | 19 | beta t1/2 | = | 1.2 | hr | ALA990662 | hr | Rattus norvegicus | |||
| 16. | ALA62811 | 19 | AUC | = | 1753 | ng.hr/ml | ALA990668 | ng.hr.mL-1 | Rattus norvegicus | |||
| 17. | ALA62811 | 19 | Cmax | = | 261 | ng/ml | ALA990666 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 18. | ALA62811 | 19 | Tmax | = | 4 | hr | ALA990664 | hr | Rattus norvegicus | |||
| 19. | ALA62811 | 19 | beta t1/2 | = | 3.8 | hr | ALA989851 | hr | Rattus norvegicus | |||
| 20. | ALA62811 | 19 | PPB | = | 61 | % | ALA989850 | % | Homo sapiens |
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