# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5200121 | rac-5b | Activity | = | 0 | % | ALA5157655 | % | Cavia porcellus | |||
2. | ALA5190238 | (1R,5S,8S)-5a | Activity | = | 0 | % | ALA5157655 | % | Cavia porcellus | |||
3. | ALA5203422 | (1S,5R,8R)-5a | Activity | = | 7 | % | ALA5157655 | % | Cavia porcellus | |||
4. | ALA5204863 | (1R,5R,7S)-4b | Activity | = | 0 | % | ALA5157655 | % | Cavia porcellus | |||
5. | ALA5185196 | (1R,5R,7S)-4a | Activity | = | 0 | % | ALA5157655 | % | Cavia porcellus | |||
6. | ALA5173028 | (1S,5S,7R)-4a | Activity | = | 0 | % | ALA5157655 | % | Cavia porcellus | |||
7. | morphine | morphine | Ki | = | 5.2 | nM | ALA5157653 | 8.28 | nM | Cavia porcellus | ||
8. | Naloxone | naloxone | Ki | = | 2.3 | nM | ALA5157653 | 8.64 | nM | Cavia porcellus | ||
9. | ALA5178401 | (1S,5S,7R)-4b | Ki | > | 1000 | nM | ALA5157653 | nM | Cavia porcellus | |||
10. | ALA5178271 | 200; MGM-16 | Ki | = | 2.1 | nM | ALA5127619 | 8.68 | nM | Cavia porcellus | ||
11. | ALA5187788 | 199; MGM-15 | Ki | = | 6.4 | nM | ALA5127619 | 8.19 | nM | Cavia porcellus | ||
12. | ALA2396991 | MGM-9 | Ki | = | 7.3 | nM | ALA5127619 | 8.14 | nM | Cavia porcellus | ||
13. | ALA5178409 | 190 | Ki | = | 11 | nM | ALA5127619 | 7.96 | nM | Cavia porcellus | ||
14. | ALA1355638 | SID50112575 | IC50 | = | 6.9 | nM | ALA5127551 | 8.16 | nM | Cavia porcellus | ||
15. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | IC50 | = | 1.41 | nM | ALA5127551 | 8.85 | nM | Cavia porcellus | ||
16. | Peanut oil hardened | DALDA | IC50 | = | 254 | nM | ALA5127551 | 6.59 | nM | Cavia porcellus | ||
17. | ALA5201627 | 116; [D-Arg2]-dermorphin (1-2) | IC50 | = | 44000 | nM | ALA5127551 | 4.36 | nM | Cavia porcellus | ||
18. | ALA1355638 | SID50112575 | IC20 | = | 21 | nM | ALA5127551 | nM | Cavia porcellus | |||
19. | ALA285479 | SID26756562 | IC50 | > | 4000 | nM | ALA5127551 | nM | Cavia porcellus | |||
20. | ALA5176903 | 118; [D-Arg2]-dermorphin (1-3) | IC50 | = | 240 | nM | ALA5127551 | 6.62 | nM | Cavia porcellus |