# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5200121 | rac-5b | Activity | = | 0 | % | ALA5157655 | % | Cavia porcellus | |||
2. | ALA5190238 | (1R,5S,8S)-5a | Activity | = | 0 | % | ALA5157655 | % | Cavia porcellus | |||
3. | ALA5203422 | (1S,5R,8R)-5a | Activity | = | 7 | % | ALA5157655 | % | Cavia porcellus | |||
4. | ALA5204863 | (1R,5R,7S)-4b | Activity | = | 0 | % | ALA5157655 | % | Cavia porcellus | |||
5. | ALA5185196 | (1R,5R,7S)-4a | Activity | = | 0 | % | ALA5157655 | % | Cavia porcellus | |||
6. | ALA5173028 | (1S,5S,7R)-4a | Activity | = | 0 | % | ALA5157655 | % | Cavia porcellus | |||
7. | morphine | morphine | Ki | = | 5.2 | nM | ALA5157653 | 8.28 | nM | Cavia porcellus | ||
8. | [³H]naloxone | naloxone | Ki | = | 2.3 | nM | ALA5157653 | 8.64 | nM | Cavia porcellus | ||
9. | ALA5178401 | (1S,5S,7R)-4b | Ki | > | 1000 | nM | ALA5157653 | nM | Cavia porcellus | |||
10. | DADLE | Tyr-D-Ala-Gly-Phe-D-Leu | Ki | = | 3.2 | nM | ALA3239406 | 8.49 | nM | Cavia porcellus | ||
11. | DADLE | Tyr-D-Ala-Gly-Phe-D-Leu | IC50 | = | 13.39 | nM | ALA3239393 | 7.87 | nM | Cavia porcellus | ||
12. | ALA120758 | 20 | IC50 | = | 2.33 | nM | ALA3239393 | 8.63 | nM | Cavia porcellus | ||
13. | ALA3233200 | 12 | IC50 | = | 0.274 | nM | ALA3239393 | 9.56 | nM | Cavia porcellus | ||
14. | ALA3233014 | 11 | IC50 | = | 2.68 | nM | ALA3239393 | 8.57 | nM | Cavia porcellus | ||
15. | ALA3233199 | 10 | IC50 | > | 10000 | nM | ALA3239393 | nM | Cavia porcellus | |||
16. | ALA3233198 | 9 | IC50 | = | 4.63 | nM | ALA3239393 | 8.33 | nM | Cavia porcellus | ||
17. | ALA3233197 | 8 | IC50 | = | 10.4 | nM | ALA3239393 | 7.98 | nM | Cavia porcellus | ||
18. | ALA3233196 | 7 | IC50 | = | 9.28 | nM | ALA3239393 | 8.03 | nM | Cavia porcellus | ||
19. | ALA3233195 | 6 | IC50 | = | 44.6 | nM | ALA3239393 | 7.35 | nM | Cavia porcellus | ||
20. | ALA3233194 | 5 | IC50 | = | 249 | nM | ALA3239393 | 6.60 | nM | Cavia porcellus |