# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4082855 | 5k | IC50 | = | 48 | uM | ALA5244931 | 4.32 | nM | Trypanosoma brucei rhodesiense | ||
2. | ALA454439 | 6d | IC50 | = | 34.2 | uM | ALA5244931 | 4.47 | nM | Trypanosoma brucei rhodesiense | ||
3. | N-(7-chloroquinolin-4-yl)ethane-1,2-diamine | 15 | IC50 | = | 125.5 | uM | ALA5244931 | nM | Trypanosoma brucei rhodesiense | |||
4. | ALA31000 | 6 | IC50 | = | 58 | uM | ALA5244931 | 4.24 | nM | Trypanosoma brucei rhodesiense | ||
5. | ALA148139 | 7 | IC50 | = | 61 | uM | ALA5244931 | 4.21 | nM | Trypanosoma brucei rhodesiense | ||
6. | ALA460418 | 6g | IC50 | = | 72 | uM | ALA5244931 | 4.14 | nM | Trypanosoma brucei rhodesiense | ||
7. | ALA528696 | TCMDC-125506 | IC50 | = | 34 | uM | ALA5244931 | 4.47 | nM | Trypanosoma brucei rhodesiense | ||
8. | ALA4247075 | FGA40 | IC50 | = | 26 | nM | ALA5244931 | 7.58 | nM | Trypanosoma brucei rhodesiense | ||
9. | ALA5275445 | Cis-79c | IC50 | = | 16.4 | nM | ALA5244931 | 7.79 | nM | Trypanosoma brucei rhodesiense | ||
10. | ALA4245127 | FGA47 | IC50 | = | 144.6 | nM | ALA5244931 | 6.84 | nM | Trypanosoma brucei rhodesiense | ||
11. | ALA4251480 | FGA44 | IC50 | = | 30.7 | nM | ALA5244931 | 7.51 | nM | Trypanosoma brucei rhodesiense | ||
12. | ALA4242650 | FGA50 | IC50 | = | 20 | uM | ALA5244931 | 4.70 | nM | Trypanosoma brucei rhodesiense | ||
13. | ALA4247075 | FGA40 | IC50 | = | 10 | uM | ALA5244931 | 5.00 | nM | Trypanosoma brucei rhodesiense | ||
14. | ALA1078675 | 3a | Ki | = | 6 | nM | ALA5244929 | 8.22 | nM | Trypanosoma brucei rhodesiense | ||
15. | K777 | 2 | Ki | = | 7 | nM | ALA5244929 | 8.15 | nM | Trypanosoma brucei rhodesiense | ||
16. | ALA5175604 | 3e | INH | = | 80 | % | ALA5163844 | % | Trypanosoma brucei rhodesiense | |||
17. | ALA5209848 | 3d | INH | = | 80 | % | ALA5163844 | % | Trypanosoma brucei rhodesiense | |||
18. | ALA5182014 | 3c | INH | = | 80 | % | ALA5163844 | % | Trypanosoma brucei rhodesiense | |||
19. | ALA5204127 | 3b | INH | = | 80 | % | ALA5163844 | % | Trypanosoma brucei rhodesiense | |||
20. | ALA5207440 | 3a | INH | = | 80 | % | ALA5163844 | % | Trypanosoma brucei rhodesiense |