| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5306285 | EUB0002235 | delta Tm Staurosporine positive control | = | 8.696 | ALA5304808 | Homo sapiens | |||||
| 2. | ALA5306285 | EUB0002235 | delta Tm | = | 0.044 | ALA5304808 | Not Active | Homo sapiens | ||||
| 3. |  ALA5308262 | EUB0002234 | delta Tm Staurosporine positive control | = | 8.696 | ALA5304704 | Homo sapiens | |||||
| 4. | ALA5308262 | EUB0002234 | delta Tm | = | 0.123 | ALA5304704 | Not Active | Homo sapiens | ||||
| 5. |  ALA5308250 | EUB0002186 | delta Tm Staurosporine positive control | = | 9.222 | ALA5304617 | Homo sapiens | |||||
| 6. | ALA5308250 | EUB0002186 | delta Tm | = | -0.389 | ALA5304617 | Not Active | Homo sapiens | ||||
| 7. |  ALA5306577 | EUB0002354 | delta Tm Staurosporine positive control | = | 9.222 | ALA5304518 | Homo sapiens | |||||
| 8. | ALA5306577 | EUB0002354 | delta Tm | = | -0.11 | ALA5304518 | Not Active | Homo sapiens | ||||
| 9. |  ALA3775317 | 31 | Activity | = | -15 | % | ALA3778581 | % | Homo sapiens | |||
| 10. |  ALA3775576 | 18 | Activity | = | -1 | % | ALA3778581 | % | Homo sapiens | |||
| 11. |  ALA3774885 | 39 | Activity | = | 2 | % | ALA3778581 | % | Homo sapiens | |||
| 12. |  ALA3758502 | 1 | INH | = | 6 | % | ALA3762703 | % | Homo sapiens | |||
| 13. |  ALA3745885 | 7ao; ON1231320 | IC50 | > | 10 | uM | ALA3748185 | nM | Homo sapiens | |||
| 14. |  ALA3746293 | 23 | INH | = | 7.2 | % | ALA3751243 | % | Homo sapiens | |||
| 15. |  A-971432 | 29; A-971432 | IC50 | > | 10 | uM | ALA3743697 | nM | Homo sapiens | |||
| 16. |  ALA3628628 | 5 | INH | = | 16.44 | % | ALA3630495 | % | Homo sapiens | |||
| 17. |  ALA3628627 | 4 | INH | = | 42.43 | % | ALA3630495 | % | Homo sapiens | |||
| 18. |  ALA166031 | 3 | INH | = | 33.81 | % | ALA3630495 | % | Homo sapiens | |||
| 19. |  ALA3623375 | 19 | IC50 | > | 10 | uM | ALA3625839 | nM | Homo sapiens | |||
| 20. |  Lorlatinib | 8k, PF-06463922 | Ki | = | 6 | nM | ALA5213171 | 8.22 | nM | Homo sapiens |
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